日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Single-cell image-based screens identify host regulators of Ebola virus infection dynamics.

基于单细胞图像的筛选方法可识别埃博拉病毒感染动态的宿主调控因子。

Carlson Rebecca J, Patten J J, Stefanakis George, Soong Brian Y, Radhakrishnan Adityanarayanan, Singh Avtar, Thakur Naveen, Sheehan Kathleen C F, Amarasinghe Gaya K, Hacohen Nir, Basler Christopher F, Leung Daisy W, Uhler Caroline, Davey Robert A, Blainey Paul C

Soluble CD4 inhibits Ebola virus infection by targeting endosomal receptor-binding site.

可溶性CD4通过靶向内体受体结合位点抑制埃博拉病毒感染

Wang Leah Liu, Keiser Patrick, Yang Derek, Seravalli Javier, Patten J J, Eaton Brett, Anderson Dirk, Liu Yi, Holbrook Michael R, Smith Amos B 3rd, Davey Robert A, Xiang Shi-Hua

Unlocking the potential of phytochemicals in inhibiting SARS-CoV-2 M(Pro) protein - an in silico and cell-based approach

利用计算机模拟和细胞方法探索植物化学物质抑制SARS-CoV-2 M(Pro)蛋白的潜力

Singh, Khushboo; Patten, J J; Dimet-Wiley, Andrea; Davey, Robert A; Watowich, Stanley J; Chandra, Amit; Leverett, Jesse

N-Substituted Pyrrole-Based Heterocycles as Broad-Spectrum Filoviral Entry Inhibitors

N-取代吡咯基杂环化合物作为广谱丝状病毒入侵抑制剂

Durante, Destiny; Bott, Ryan; Cooper, Laura; Owen, Callum; Morsheimer, Kimberly M; Patten, J J; Zielinski, Christian; Peet, Norton P; Davey, Robert A; Gaisina, Irina N; Rong, Lijun; Moore, Terry W

Amidino-rocaglates (ADRs), a class of synthetic rocaglates, are potent inhibitors of SARS-CoV-2 replication through inhibition of viral protein synthesis.

脒基罗卡格列酸酯(ADRs)是一类合成罗卡格列酸酯,可通过抑制病毒蛋白合成来有效抑制SARS-CoV-2复制

Keiser Patrick T, Zhang Wenhan, Ricca Michael, Wacquiez Alan, Grimins Autumn, Cencic Regina, Patten J J, Shah Pranav, Padilha Elias, Connor John H, Pelletier Jerry, Lyons Shawn M, Saeed Mohsan, Brown Lauren E, Porco John A Jr, Davey Robert A

Anti-SARS-CoV-2 activity of targeted kinase inhibitors: Repurposing clinically available drugs for COVID-19 therapy

靶向激酶抑制剂的抗SARS-CoV-2活性:将临床可用药物重新用于COVID-19治疗

Boytz, RuthMabel; Słabicki, Mikołaj; Ramaswamy, Sita; Patten, J J; Zou, Charles; Meng, Chengcheng; Hurst, Brett L; Wang, Jinhua; Nowak, Radosław P; Yang, Priscilla L; Sattler, Martin; Stone, Richard M; Griffin, James D; Gray, Nathanael S; Gummuluru, Suryaram; Davey, Robert A; Weisberg, Ellen

Network medicine framework for identifying drug-repurposing opportunities for COVID-19

利用网络医学框架识别新冠肺炎药物再利用机会

Morselli Gysi, Deisy; do Valle, Ítalo; Zitnik, Marinka; Ameli, Asher; Gan, Xiao; Varol, Onur; Ghiassian, Susan Dina; Patten, J J; Davey, Robert A; Loscalzo, Joseph; Barabási, Albert-László

A multi-pronged approach targeting SARS-CoV-2 proteins using ultra-large virtual screening

利用超大规模虚拟筛选技术,采用多管齐下的方法靶向SARS-CoV-2蛋白

Gorgulla, Christoph; Padmanabha Das, Krishna M; Leigh, Kendra E; Cespugli, Marco; Fischer, Patrick D; Wang, Zi-Fu; Tesseyre, Guilhem; Pandita, Shreya; Shnapir, Alec; Calderaio, Anthony; Gechev, Minko; Rose, Alexander; Lewis, Noam; Hutcheson, Colin; Yaffe, Erez; Luxenburg, Roni; Herce, Henry D; Durmaz, Vedat; Halazonetis, Thanos D; Fackeldey, Konstantin; Patten, J J; Chuprina, Alexander; Dziuba, Igor; Plekhova, Alla; Moroz, Yurii; Radchenko, Dmytro; Tarkhanova, Olga; Yavnyuk, Irina; Gruber, Christian; Yust, Ryan; Payne, Dave; Näär, Anders M; Namchuk, Mark N; Davey, Robert A; Wagner, Gerhard; Kinney, Jamie; Arthanari, Haribabu

Identification of filovirus entry inhibitors targeting the endosomal receptor NPC1 binding site

鉴定靶向内体受体NPC1结合位点的丝状病毒进入抑制剂

Wang, Leah Liu; Palermo, Nicholas; Estrada, Leslie; Thompson, Colton; Patten, J J; Anantpadma, Manu; Davey, Robert A; Xiang, Shi-Hua