日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nav1.8 mediates peripheral-to-central nociceptive transmission independently of central presynaptic mechanisms in human DRG-spinal cord circuits

在人类背根神经节-脊髓回路中,Nav1.8 介导外周到中枢的伤害性感受传递,且该过程独立于中枢突触前机制。

Palomino, Seph M; Gabriel, Katherin A; Koduri, Ashwin; Khan, Ibrahim; Syed A, Rahman; Horton, Peter; Khan, Tariq; Cervantes, Anna; Funk, Geoffrey; Shiers, Stephanie; Price, Theodore J; Patwardhan, Amol

The conotoxin Contulakin-G reverses hypersensitivity observed in rodent models of cancer-induced bone pain without inducing tolerance or motor disturbance.

芋螺毒素 Contulakin-G 可逆转啮齿动物癌症诱发骨痛模型中观察到的过敏反应,而不会引起耐受性或运动障碍

Martin Laurent F, Almuslim Moyad, Ismail Khaled A, Ibrahim Mohab M, Moutal Aubin, Cheng Kevin, Stratton Harrison J, Price Theodore J, Vanderah Todd W, Olivera Baldomero M, Khanna Rajesh, Patwardhan Amol

Cone snail venom-inspired somatostatin receptor 4 (SSTR(4)) agonists as new drug leads for peripheral pain

锥螺毒液启发的生长抑素受体4 (SSTR(4))激动剂作为治疗外周疼痛的新药先导化合物

Bjørn-Yoshimoto, Walden E; Ramiro, Iris Bea L; Koch, Thomas Lund; Engholm, Ebbe; Yeung, Ho Yan; Sørensen, Kasper K; Goddard, Carolyn M; Jensen, Kathrine L; Smith, Nicholas A; Martin, Laurent F; Smith, Brian J; Madsen, Kenneth L; Jensen, Knud J; Patwardhan, Amol; Safavi-Hemami, Helena

Genetic editing of primary human dorsal root ganglion neurons using CRISPR-Cas9.

利用 CRISPR-Cas9 对人类原代背根神经节神经元进行基因编辑

Palomino Seph M, Gabriel Katherin A, Mwirigi Juliet M, Cervantes Anna, Horton Peter, Funk Geoffrey, Moutal Aubin, Martin Laurent F, Khanna Rajesh, Price Theodore J, Patwardhan Amol

Expansion of OSMR expression and signaling in the human dorsal root ganglion links OSM to neuropathic pain

人类背根神经节中OSMR表达和信号传导的扩展将OSM与神经性疼痛联系起来

Mwirigi, Juliet M; Sankaranarayanan, Ishwarya; Tavares-Ferreira, Diana; Gabriel, Katherin A; Palomino, Seph; Li, Yan; Uhelski, Megan L; Shiers, Stephanie; Franco-Enzástiga, Úrzula; Wangzhou, Andi; Lesnak, Joseph B; Bandaru, Samhita; Shrivastava, Aishni; Inturi, Nikhil; Albrecht, Phillip J; Dockum, Marilyn; Cervantes, Anna M; Horton, Peter; Funk, Geoffrey; North, Robert Y; Tatsui, Claudio Esteves; Corrales, German; Yousuf, Muhammad Saad; Curatolo, Michele; Gereau, Robert W; Patwardhan, Amol; Dussor, Gregory; Dougherty, Patrick M; Rice, Frank L; Price, Theodore J

Dantrolene for the Treatment of Chronic Inflammatory Demyelinating Polyneuropathy-Induced Painful Muscle Spasms: A Case Report

丹曲林治疗慢性炎症性脱髓鞘性多发性神经病引起的疼痛性肌肉痉挛:病例报告

Martins, Yuri Chaves; Jain, Sejal V; Patwardhan, Amol M

A molecular map of the human spinal dorsal and ventral horn defines arrangement of neuronal types and glial sex differences

人类脊髓背角和腹角的分子图谱揭示了神经元类型的排列以及神经胶质细胞的性别差异。

Gabriel, Katherin A; Davis, Olivia C; Palomino, Seph M; Ishishita, Satoshi; Poldsam, Helen; Brandon, Jane M; Inturi, Nikhil N; Mydugolam, Hemanth; Khan, Ibrahim O; Selvakumaran, Nethra; Shiers, Stephanie; Yousuf, Muhammad Saad; Vines, Erin; Horton, Peter; Khan, Tariq; Cervantes, Anna; Reese, Jeffrey C; Patwardhan, Amol; Dussor, Gregory; Meyers, Eric; Tavares-Ferreira, Diana; Pool, Allan-Hermann; Price, Theodore J

C2230, a preferential use- and state-dependent CaV2.2 channel blocker, mitigates pain behaviors across multiple pain models.

C2230 是一种优先使用和状态依赖的 CaV2.2 通道阻滞剂,可减轻多种疼痛模型中的疼痛行为

Tang Cheng, Gomez Kimberly, Chen Yan, Allen Heather N, Hestehave Sara, Rodríguez-Palma Erick J, Loya-Lopez Santiago, Calderon-Rivera Aida, Duran Paz, Nelson Tyler S, Kanumuri Siva Rama Raju, Shah Bijal, Panigrahi Nihar R, Perez-Miller Samantha, Schackmuth Morgan K, Ruparel Shivani, Patwardhan Amol, Price Theodore J, Arora Paramjit S, Sharma Ravindra K, Sharma Abhisheak, Yu Jie, Korczeniewska Olga A, Khanna Rajesh

Chronic pain recruits hypothalamic dynorphin/kappa opioid receptor signalling to promote wakefulness and vigilance

慢性疼痛会激活下丘脑强啡肽/κ阿片受体信号通路,从而促进觉醒和警觉。

Ito, Hisakatsu; Navratilova, Edita; Vagnerova, Barbora; Watanabe, Moe; Kopruszinski, Carol; Moreira de Souza, Luiz H; Yue, Xu; Ikegami, Daigo; Moutal, Aubin; Patwardhan, Amol; Khanna, Rajesh; Yamazaki, Mitsuaki; Guerrero, Miguel; Rosen, Hugh; Roberts, Ed; Neugebauer, Volker; Dodick, David W; Porreca, Frank

Oral Cancer Pain Includes Thermal Allodynia That May Be Attenuated by Chronic Alcohol Consumption

口腔癌疼痛包括热痛觉过敏,这种疼痛可能会因长期饮酒而减轻。

Gonzales, Cara B; De La Chapa, Jorge J; Patwardhan, Amol M; Hargreaves, Kenneth M