日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulation of SF3B1 in the pre-mRNA spliceosome induces a RIG-I-dependent type I IFN response

前体mRNA剪接体中SF3B1的调控可诱导RIG-I依赖的I型干扰素反应。

Aaron Y Chang ,Yu Jerry Zhou ,Sharanya Iyengar ,Piotr W Pobiarzyn ,Pavel Tishchenko ,Kesha M Shah ,Heather Wheeler ,Yue-Ming Wang ,Paula M Loria ,Frank Loganzo ,Seng-Ryong Woo

Selective stalling of human translation through small-molecule engagement of the ribosome nascent chain

通过小分子参与核糖体新生链选择性停止人类翻译

Nathanael G Lintner, Kim F McClure, Donna Petersen, Allyn T Londregan, David W Piotrowski, Liuqing Wei, Jun Xiao, Michael Bolt, Paula M Loria, Bruce Maguire, Kieran F Geoghegan, Austin Huang, Tim Rolph, Spiros Liras, Jennifer A Doudna, Robert G Dullea, Jamie H D Cate

Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate

发现 PF-5190457,一种强效、选择性、口服生物可利用的生长素释放肽受体反向激动剂临床候选药物

Samit K Bhattacharya, Kim Andrews, Ramsay Beveridge, Kimberly O Cameron, Chiliu Chen, Matthew Dunn, Dilinie Fernando, Hua Gao, David Hepworth, V Margaret Jackson, Vishal Khot, Jimmy Kong, Rachel E Kosa, Kimberly Lapham, Paula M Loria, Allyn T Londregan, Kim F McClure, Suvi T M Orr, Jigna Patel, Coli

Antibody-directed myostatin inhibition improves diaphragm pathology in young but not adult dystrophic mdx mice

抗体导向的肌生长抑制素抑制可改善年轻但成年营养不良 mdx 小鼠的膈肌病理

Kate T Murphy, James G Ryall, Sarah M Snell, Lawrence Nair, René Koopman, Philip A Krasney, Chikwendu Ibebunjo, Kathryn S Holden, Paula M Loria, Christopher T Salatto, Gordon S Lynch