Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate
发现 PF-5190457,一种强效、选择性、口服生物可利用的生长素释放肽受体反向激动剂临床候选药物
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/ml400473x
Samit K Bhattacharya, Kim Andrews, Ramsay Beveridge, Kimberly O Cameron, Chiliu Chen, Matthew Dunn, Dilinie Fernando, Hua Gao, David Hepworth, V Margaret Jackson, Vishal Khot, Jimmy Kong, Rachel E Kosa, Kimberly Lapham, Paula M Loria, Allyn T Londregan, Kim F McClure, Suvi T M Orr, Jigna Patel, Coli