日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A multiplex method for rapidly identifying viral protease inhibitors

一种快速鉴定病毒蛋白酶抑制剂的多重检测方法

Seo Jung Hong # ,Samuel J Resnick # ,Sho Iketani # ,Ji Won Cha ,Benjamin Alexander Albert ,Christopher T Fazekas ,Ching-Wen Chang ,Hengrui Liu ,Shlomi Dagan ,Michael R Abagyan ,Pavla Fajtová ,Bruce Culbertson ,Brooklyn Brace ,Eswar R Reddem ,Farhad Forouhar ,J Fraser Glickman ,James M Balkovec ,Brent R Stockwell ,Lawrence Shapiro ,Anthony J O'Donoghue ,Yosef Sabo ,Joel S Freundlich ,David D Ho ,Alejandro Chavez

Nature-Inspired Gallinamides Are Potent Antischistosomal Agents: Inhibition of the Cathepsin B1 Protease Target and Binding Mode Analysis

源自自然的加林酰胺是有效的抗血吸虫剂:抑制组织蛋白酶 B1 蛋白酶靶标和结合模式分析

Petra Spiwoková, Martin Horn, Jindřich Fanfrlík, Adéla Jílková, Pavla Fajtová, Adrian Leontovyč, Radka Houštecká, Lucia Bieliková, Jiří Brynda, Marta Chanová, Helena Mertlíková-Kaiserová, Eduardo J E Caro-Diaz, Jehad Almaliti, Nelly El-Sakkary, William H Gerwick, Conor R Caffrey, Michael Mareš

Evaluating Antimalarial Proteasome Inhibitors for Efficacy in Babesia Blood Stage Cultures

评估抗疟蛋白酶体抑制剂对巴贝斯虫血液阶段培养物的疗效

Luïse Robbertse, Pavla Fajtová, Pavla Šnebergerová, Marie Jalovecká, Viktoriya Levytska, Elany Barbosa da Silva, Vandna Sharma, Petr Pachl, Jehad Almaliti, Momen Al-Hindy, William H Gerwick, Evžen Bouřa, Anthony J O'Donoghue, Daniel Sojka

Development of subunit selective proteasome substrates for Schistosoma species

血吸虫亚基选择性蛋白酶体底物的开发

Zhenze Jiang, Elany B Silva, Chenxi Liu, Pavla Fajtová, Lawrence J Liu, Nelly El-Sakkary, Danielle E Skinner, Ali Syed, Steven C Wang, Conor R Caffrey, Anthony J O'Donoghue

Large library docking for novel SARS-CoV-2 main protease non-covalent and covalent inhibitors

新型 SARS-CoV-2 主蛋白酶非共价和共价抑制剂的大型文库对接

Elissa A Fink, Conner Bardine, Stefan Gahbauer, Isha Singh, Tyler C Detomasi, Kris White, Shuo Gu, Xiaobo Wan, Jun Chen, Beatrice Ary, Isabella Glenn, Joseph O'Connell, Henry O'Donnell, Pavla Fajtová, Jiankun Lyu, Seth Vigneron, Nicholas J Young, Ivan S Kondratov, Arghavan Alisoltani, Lacy M Simons,

Development of Potent and Highly Selective Epoxyketone-Based Plasmodium Proteasome Inhibitors

开发强效、高选择性的基于环氧酮的疟原虫蛋白酶体抑制剂

Jehad Almaliti, Pavla Fajtová, Jaeson Calla, Gregory M LaMonte, Mudong Feng, Frances Rocamora, Sabine Ottilie, Evgenia Glukhov, Evzen Boura, Raymond T Suhandynata, Jeremiah D Momper, Michael K Gilson, Elizabeth A Winzeler, William H Gerwick, Anthony J O'Donoghue

Native metabolomics identifies the rivulariapeptolide family of protease inhibitors

天然代谢组学鉴定了 rivulariapeptolide 家族的蛋白酶抑制剂

Raphael Reher, Allegra T Aron, Pavla Fajtová, Paolo Stincone, Berenike Wagner, Alicia I Pérez-Lorente, Chenxi Liu, Ido Y Ben Shalom, Wout Bittremieux, Mingxun Wang, Kyowon Jeong, Marie L Matos-Hernandez, Kelsey L Alexander, Eduardo J Caro-Diaz, C Benjamin Naman, J H William Scanlan, Phil M M Hochban

Potent Anti-SARS-CoV-2 Activity by the Natural Product Gallinamide A and Analogues via Inhibition of Cathepsin L

天然产物 Gallinamide A 及其类似物通过抑制组织蛋白酶 L 发挥强效抗 SARS-CoV-2 活性

Anneliese S Ashhurst, Arthur H Tang, Pavla Fajtová, Michael C Yoon, Anupriya Aggarwal, Max J Bedding, Alexander Stoye, Laura Beretta, Dustin Pwee, Aleksandra Drelich, Danielle Skinner, Linfeng Li, Thomas D Meek, James H McKerrow, Vivian Hook, Chien-Te Tseng, Mark Larance, Stuart Turville, William H

Discovery of Triple Inhibitors of Both SARS-CoV-2 Proteases and Human Cathepsin L

发现 SARS-CoV-2 蛋白酶和人类组织蛋白酶 L 的三重抑制剂

Ittipat Meewan, Jacob Kattoula, Julius Y Kattoula, Danielle Skinner, Pavla Fajtová, Miriam A Giardini, Brendon Woodworth, James H McKerrow, Jair Lage de Siqueira-Neto, Anthony J O'Donoghue, Ruben Abagyan

Activatable Carbocyanine Dimers for Photoacoustic and Fluorescent Detection of Protease Activity

可激活的碳菁二聚体用于光声和荧光检测蛋白酶活性

Colman Moore, Raina M Borum, Yash Mantri, Ming Xu, Pavla Fajtová, Anthony J O'Donoghue, Jesse V Jokerst