日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proximity-Induced Rewiring of Oncogenic Kinase Triggers Apoptosis

邻近诱导的致癌激酶重编程触发细胞凋亡

Merz, Manuel L; Shoba, Veronika M; Pergu, Rajaiah; Severance, Zachary C; Munkanatta Godage, Dhanushka N P; Deb, Arghya; Kwok, Hui Si; Singh, Prashant; Singh, Sameek; Allen, Jonathan B; Tian, Wenzhi; Gosavi, Pallavi M; Chaudhary, Santosh K; Anokhina, Viktoriya; Weisberg, Ellen L; Payne, N Connor; He, Yao; Dhaliwal, Rohil; Osadchey, Reilly; Shekhar, Mrinal; Mazitschek, Ralph; Rees, Matthew G; Roth, Jennifer A; Cui, Qiang; Griffin, James D; Liau, Brian B; Choudhary, Amit

The contribution of cyclic imide stereoisomers on cereblon-dependent activity

环状酰亚胺立体异构体对脑蛋白依赖性活性的影响

Amako, Yuka; Ichikawa, Saki; Lloyd, Hannah C; Payne, N Connor; Lin, Zhi; Boghossian, Andrew S; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Zhu, Qian; Budnik, Bogdan; Mazitschek, Ralph; Woo, Christina M

Revisiting the Plasmodium falciparum druggable genome using predicted structures and data mining

利用预测结构和数据挖掘技术重新审视恶性疟原虫可药物靶向基因组

Godinez-Macias, Karla P; Chen, Daisy; Wallis, J Lincoln; Siegel, Miles G; Adam, Anna; Bopp, Selina; Carolino, Krypton; Coulson, Lauren B; Durst, Greg; Thathy, Vandana; Esherick, Lisl; Farringer, Madeline A; Flannery, Erika L; Forte, Barbara; Liu, Tiqing; Godoy Magalhaes, Luma; Gupta, Anil K; Istvan, Eva S; Jiang, Tiantian; Kumpornsin, Krittikorn; Lobb, Karen; McLean, Kyle J; Moura, Igor M R; Okombo, John; Payne, N Connor; Plater, Andrew; Rao, Srinivasa P S; Siqueira-Neto, Jair L; Somsen, Bente A; Summers, Robert L; Zhang, Rumin; Gilson, Michael K; Gamo, Francisco-Javier; Campo, Brice; Baragaña, Beatriz; Duffy, James; Gilbert, Ian H; Lukens, Amanda K; Dechering, Koen J; Niles, Jacquin C; McNamara, Case W; Cheng, Xiu; Birkholtz, Lyn-Marie; Bronkhorst, Alfred W; Fidock, David A; Wirth, Dyann F; Goldberg, Daniel E; Lee, Marcus C S; Winzeler, Elizabeth A

A method for the detection and enrichment of endogenous cereblon substrates.

一种检测和富集内源性 cereblon 底物的方法

Lloyd Hannah C, Li Yuli, Payne N Connor, Zhao Zhenguang, Xu Wenqing, Kroupova Alena, Zollman David, Long Tengfang, Kabir Farah, Chen Mei, Freeman Rebecca, Feng Ethan Yang, Xi Sarah, Hsu Ya-Chieh, Ciulli Alessio, Mazitschek Ralph, Woo Christina M

Phosphorylation-inducing chimera rewires oncogenic kinase to trigger apoptosis.

磷酸化诱导嵌合体重塑致癌激酶以触发细胞凋亡

Merz Manuel L, Shoba Veronika M, Pergu Rajaiah, Severance Zachary C, Munkanatta Godage Dhanushka N P, Deb Arghya, Kwok Hui Si, Singh Prashant, Singh Sameek, Allen Jonathan B, Tian Wenzhi, Gosavi Pallavi M, Chaudhary Santosh K, Anokhina Viktoriya, Weisberg Ellen L, Payne N Connor, He Yao, Osadchey Reilly, Shekhar Mrinal, Mazitschek Ralph, Rees Matthew G, Roth Jennifer A, Cui Qiang, Griffin James D, Liau Brian B, Choudhary Amit

Inhibiting the Keap1/Nrf2 Protein-Protein Interaction with Protein-Like Polymers

利用类蛋白聚合物抑制Keap1/Nrf2蛋白-蛋白相互作用

Carrow, Kendal P; Hamilton, Haylee L; Hopps, Madeline P; Li, Yang; Qiao, Baofu; Payne, N Connor; Thompson, Matthew P; Zhang, Xiaoyu; Magassa, Assa; Fattah, Mara; Agarwal, Shivangi; Vincent, Michael P; Buyanova, Marina; Bertin, Paul A; Mazitschek, Ralph; Olvera de la Cruz, Monica; Johnson, Delinda A; Johnson, Jeffrey A; Gianneschi, Nathan C

Identification of a Polypeptide Inhibitor of O-GlcNAc Transferase with Picomolar Affinity

鉴定出一种对 O-GlcNAc 转移酶具有皮摩尔级亲和力的多肽抑制剂

Hammel, Forrest A; Payne, N Connor; Marando, Victoria M; Mazitschek, Ralph; Walker, Suzanne

Correction: Prolyl-tRNA synthetase as a novel therapeutic target in multiple myeloma

更正:脯氨酰-tRNA合成酶作为多发性骨髓瘤的新型治疗靶点

Kurata, Keiji; James-Bott, Anna; Tye, Mark A; Yamamoto, Leona; Samur, Mehmet K; Tai, Yu-Tzu; Dunford, James; Johansson, Catrine; Senbabaoglu, Filiz; Philpott, Martin; Palmer, Charlotte; Ramasamy, Karthik; Gooding, Sarah; Smilova, Mihaela; Gaeta, Giorgia; Guo, Manman; Christianson, John C; Payne, N Connor; Singh, Kritika; Karagoz, Kubra; Stokes, Matthew E; Ortiz, Maria; Hagner, Patrick; Thakurta, Anjan; Cribbs, Adam; Mazitschek, Ralph; Hideshima, Teru; Anderson, Kenneth C; Oppermann, Udo

Structural and biochemical characterization establishes a detailed understanding of KEAP1-CUL3 complex assembly.

结构和生化表征建立了对 KEAP1-CUL3 复合物组装的详细了解

Adamson Roslin J, Payne N Connor, Bartual Sergio G, Mazitschek Ralph, Bullock Alex N

Can dimedone be used to study selenoproteins? An investigation into the reactivity of dimedone toward oxidized forms of selenocysteine

二甲酮可用于研究硒蛋白吗?一项关于二甲酮与硒代半胱氨酸氧化形式反应性的研究

Payne, N Connor; Barber, Drew R; Ruggles, Erik L; Hondal, Robert J