日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Plasmodiumfalciparum protein kinase 6 and hemozoin formation are inhibited by a type II human kinase inhibitor exhibiting antimalarial activity

一种具有抗疟活性的II型人激酶抑制剂可抑制恶性疟原虫蛋白激酶6和血红素的形成。

Flore Nardella ,Tiantian Jiang ,Lushun Wang ,Monica J Bohmer ,Subhoja Chakraborty ,John Okombo ,Jaeson Calla ,Tatiane Macedo Silva ,Samuel Pazicky ,Jianwei Che ,Jin Jeon ,Evie Vincent ,Nonlawat Boonyalai ,Rachael Coyle ,Mairi J Buchanan ,Samuel Schaefer ,Daisy Chen ,Amaan Khan ,Emily Mayville ,Mariana Laureano De Souza ,Mayland Treat ,Jordan Charlton ,Patrick K Tumwebaze ,Seth Tjia ,Lukas Montejo ,Karen Cover ,Philip J Rosenthal ,Roland A Cooper ,Zbynek Bozdech ,Marcus C S Lee ,Ratna Chakrabarti ,Sanjay A Desai ,David A Fidock ,Jinhua Wang ,Nathanael S Gray ,Elizabeth A Winzeler ,Debopam Chakrabarti

Characterizing the quick-killing mechanism of action of azithromycin analogs against malaria parasites

阐明阿奇霉素类似物对疟原虫的快速杀灭机制

Mao, Emma Y; Nguyen, William; Jana, Gouranga P; Maity, Bikash C; Pazicky, Samuel; Giannangelo, Carlo; Reader, Janette; Famodimu, Mufuliat T; Birkholtz, Lyn-Marie; Delves, Michael J; Creek, Darren J; Bozdech, Zbynek; Laleu, Benoît; Burrows, Jeremy N; Sleebs, Brad E; Gancheva, Maria R; Wilson, Danny W

Structure of the human NK cell NKR-P1:LLT1 receptor:ligand complex reveals clustering in the immune synapse

人类 NK 细胞 NKR-P1:LLT1 受体:配体复合物的结构揭示了免疫突触中的聚集

Jan Bláha, Tereza Skálová, Barbora Kalousková, Ondřej Skořepa, Denis Cmunt, Valéria Grobárová, Samuel Pazicky, Edita Poláchová, Celeste Abreu, Jan Stránský, Tomáš Kovaľ, Jarmila Dušková, Yuguang Zhao, Karl Harlos, Jindřich Hašek, Jan Dohnálek, Ondřej Vaněk

Impact of distant peptide substrate residues on enzymatic activity of SlyD

远端肽底物残基对SlyD酶活性的影响

Pazicky, Samuel; Werle, Anna-Leoni A; Lei, Jian; Löw, Christian; Weininger, Ulrich

N-terminal phosphorylation regulates the activity of glycogen synthase kinase 3 from Plasmodium falciparum

N端磷酸化调节恶性疟原虫糖原合酶激酶3的活性

Samuel Pazicky, Arne Alder, Haydyn Mertens, Dmitri Svergun, Tim Gilberger, Christian Löw

Functional inactivation of Plasmodium falciparum glycogen synthase kinase GSK3 modulates erythrocyte invasion and blocks gametocyte maturation

恶性疟原虫糖原合成酶激酶GSK3的功能失活会调节红细胞入侵并阻断配子体成熟。

Alder, Arne; Wilcke, Louisa; Pietsch, Emma; von Thien, Heidrun; Pazicky, Samuel; Löw, Christian; Mesen-Ramirez, Paolo; Bachmann, Anna; Burda, Paul-Christian; Kunick, Conrad; Sondermann, Holger; Wilson, Danny; Gilberger, Tim-Wolf

Structural role of essential light chains in the apicomplexan glideosome

顶复门滑行体中必需轻链的结构作用

Pazicky, Samuel; Dhamotharan, Karthikeyan; Kaszuba, Karol; Mertens, Haydyn D T; Gilberger, Tim; Svergun, Dmitri; Kosinski, Jan; Weininger, Ulrich; Löw, Christian

Natural Killer Cell Activation Receptor NKp30 Oligomerization Depends on Its N-Glycosylation

自然杀伤细胞活化受体 NKp30 寡聚化依赖于其 N-糖基化

Ondřej Skořepa, Samuel Pazicky, Barbora Kalousková, Jan Bláha, Celeste Abreu, Tomáš Ječmen, Michal Rosůlek, Alexander Fish, Arthur Sedivy, Karl Harlos, Jan Dohnálek, Tereza Skálová, Ondřej Vaněk