日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical and first-in-human of purinostat mesylate, a novel selective HDAC I/IIb inhibitor, in relapsed/refractory multiple myeloma and lymphoma.

普利诺他甲磺酸盐(一种新型选择性 HDAC I/IIb 抑制剂)在复发/难治性多发性骨髓瘤和淋巴瘤中的临床前和首次人体试验

Yang Linyu, Qiu Qiang, Wang Jie, Wen Yi, Li He, Liang Rui, Feng Yunyu, Wang Fang, Lin Xiaojing, Tang Minghai, Yang Jianhong, Pei Heying, Zhao Peng, Wang Jishi, Xiang Jin, Miao Jia, Zheng Li, Tan Ke, Wang Yongsheng, Hu Yiguo, Chen Lijuan, Zhao Weili, Niu Ting

Identification of a ligand-binding site on tubulin mediating the tubulin-RB3 interaction

鉴定出微管蛋白上介导微管蛋白-RB3相互作用的配体结合位点。

Li, Yong; Zhang, Chufeng; Tang, Dongmei; Wang, Tao; Yan, Wei; Yang, Linyu; Bai, Peng; Tang, Minghai; Pei, Heying; Chen, Lijuan; Chen, Qiang; Yang, Jianhong

Correction to: Preclinical studies of Flonoltinib Maleate, a novel JAK2/FLT3 inhibitor, in treatment of JAK2(V617F)-induced myeloproliferative neoplasms

更正:新型 JAK2/FLT3 抑制剂马来酸氟诺替尼治疗 JAK2(V617F) 诱导的骨髓增生性肿瘤的临床前研究

Hu, Mengshi; Yang, Tao; Yang, Linyu; Niu, Lu; Zhu, Jinbing; Zhao, Ailin; Shi, Mingsong; Yuan, Xue; Tang, Minghai; Yang, Jianhong; Pei, Heying; Yang, Zhuang; Chen, Qiang; Ye, Haoyu; Niu, Ting; Chen, Lijuan

Therapeutic efficacy of an injectable formulation of purinostat mesylate in SU-DHL-6 tumour model

注射用普利诺司他甲磺酸盐制剂在SU-DHL-6肿瘤模型中的治疗效果

Zhu, Zejiang; Wen, Jiaolin; Xu, Yaohui; Pei, Heying; Li, Dan; Tang, Minghai; Bai, Peng; He, Jun; Yang, Zhuang; Chen, Lijuan

Cevipabulin-tubulin complex reveals a novel agent binding site on α-tubulin with tubulin degradation effect

Cevipabulin-微管蛋白复合物揭示了α-微管蛋白上一个新的药物结合位点,并具有微管蛋白降解作用。

Yang, Jianhong; Yu, Yamei; Li, Yong; Yan, Wei; Ye, Haoyu; Niu, Lu; Tang, Minghai; Wang, Zhoufeng; Yang, Zhuang; Pei, Heying; Wei, Haoche; Zhao, Min; Wen, Jiaolin; Yang, Linyu; Ouyang, Liang; Wei, Yuquan; Chen, Qiang; Li, Weimin; Chen, Lijuan

Correction: Non-toxic dose of liposomal honokiol suppresses metastasis of hepatocellular carcinoma through destabilizing EGFR and inhibiting the downstream pathways

更正:无毒剂量的脂质体厚朴酚通过破坏 EGFR 稳定性并抑制下游通路来抑制肝细胞癌转移。

Yang, Jianhong; Pei, Heying; Luo, Hong; Fu, Afu; Yang, Hansuo; Hu, Jia; Zhao, Chengjian; Chai, LuLu; Chen, Xiang; Shao, Ximing; Wang, Chunyu; Wu, Wenshuang; Wan, Li; Ye, Haoyu; Qiu, Qiang; Peng, Aihua; Wei, Yuquan; Yang, Li; Chen, Lijuan

SKLB023 protects mice against acute liver injury by inhibiting proinflammatory cytokine production in both T cells and macrophages

SKLB023 通过抑制 T 细胞和巨噬细胞中促炎细胞因子的产生,保护小鼠免受急性肝损伤。

Yu, Jia; Liu, Lili; Zhang, Huiming; Wu, Yating; Pei, Heying; Ma, Liang; Xiong, Anwen; Xie, Caifeng