日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and Synthesis of Novel Candidate CK1δ Proteolysis Targeting Chimeras (PROTACs).

新型候选CK1δ蛋白水解靶向嵌合体(PROTACs)的设计与合成。

Arnold Malte, Thompson Temi, Glennie Lorraine, Hollnagel Mattes, Sapkota Gopal, Peifer Christian

Addressing the Intracellular Vestibule of the Plasmodial Lactate Transporter PfFNT by p-Substituted Inhibitors Amplifies In Vitro Activity

通过对质粒乳酸转运蛋白 PfFNT 的细胞内前庭进行 p-取代抑制剂处理,可增强其体外活性。

Nerlich, Cornelius; Tiedjens, Finn; Hertel, Robin; Henke, Björn; Häuer, Susan; Panitzsch, Lea S; Hansen, Kerrin; Franck, Ole; Mete, Antonio; Leroy, Didier; Schade, Dennis; Peifer, Christian; Hannus, Stefan; Becker, Frank; Wittlin, Sergio; Spielmann, Tobias; Beitz, Eric

Novel Henna-Related Naphthazarine Photosensitizers for an Effective Photodynamic Therapy of Onychomycosis

新型指甲花相关萘并扎林类光敏剂用于有效治疗甲癣的光动力疗法

Baier, Joana; Jansen, Björn; Wenzel-Storjohann, Arlette; Tasdemir, Deniz; Peifer, Christian

Photopharmacological Applications for Cherenkov Radiation Generated by Clinically Used Radionuclides

临床使用放射性核素产生的切伦科夫辐射的光药理学应用

Krebs, Melanie; Döbber, Alexander; Rodat, Theo; Lützen, Ulf; Zhao, Yi; Zuhayra, Maaz; Peifer, Christian

Photoswitchable Azo- and Diazocine-Functionalized Derivatives of the VEGFR-2 Inhibitor Axitinib

VEGFR-2抑制剂阿昔替尼的光开关偶氮和二氮杂辛功能化衍生物

Heintze, Linda; Schmidt, Dorian; Rodat, Theo; Witt, Lydia; Ewert, Julia; Kriegs, Malte; Herges, Rainer; Peifer, Christian

New Discorhabdin Alkaloids from the Antarctic Deep-Sea Sponge Latrunculia biformis

来自南极深海海绵 Latrunculia biformis 的新 Discorhabdin 生物碱

Li, Fengjie; Peifer, Christian; Janussen, Dorte; Tasdemir, Deniz

Targeted Isolation of Tsitsikammamines from the Antarctic Deep-Sea Sponge Latrunculia biformis by Molecular Networking and Anticancer Activity

利用分子网络技术从南极深海海绵双形拉特伦库利亚(Latrunculia biformis)中靶向分离齐齐卡胺类化合物及其抗癌活性

Li, Fengjie; Janussen, Dorte; Peifer, Christian; Pérez-Victoria, Ignacio; Tasdemir, Deniz

A CK1 FRET biosensor reveals that DDX3X is an essential activator of CK1ε.

CK1 FRET 生物传感器显示 DDX3X 是 CK1α 的重要激活剂

Dolde Christine, Bischof Joachim, Grüter Simon, Montada Anna, Halekotte Jakob, Peifer Christian, Kalbacher Hubert, Baumann Ulrich, Knippschild Uwe, Suter Beat

Development and Biological Evaluation of a Photoactivatable Small Molecule Microtubule-Targeting Agent

光活化小分子微管靶向剂的开发和生物学评价

Döbber, Alexander; Phoa, Athena F; Abbassi, Ramzi H; Stringer, Brett W; Day, Bryan W; Johns, Terrance G; Abadleh, Mohammed; Peifer, Christian; Munoz, Lenka

Photoactivatable Caged Prodrugs of VEGFR-2 Kinase Inhibitors

光活化笼状VEGFR-2激酶抑制剂前药

Pinchuk, Boris; Horbert, Rebecca; Döbber, Alexander; Kuhl, Lydia; Peifer, Christian