日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Next-Generation GLUT Inhibitors: Lactone to Lactam Conversion in Rapaglutin A Confers Resistance to Plasma Esterases

新一代 GLUT 抑制剂:雷帕格鲁汀 A 中内酯向内酰胺的转化赋予其对血浆酯酶的抵抗力

Rao, A V Subba; Kotlyar, Marnie; Peng, Hanjing; Liu, Jun O

Identification of Rapaglutin E as an Isoform-Specific Inhibitor of Glucose Transporter 1

雷帕格鲁汀E被鉴定为葡萄糖转运蛋白1的同工型特异性抑制剂

Kotlyar, Marnie; Guo, Zufeng; Rao, A V Subba; Peng, Hanjing; Wang, Jingxin; Ma, Zhongnan; Schiene-Fischer, Cordelia; Fischer, Gunter; Liu, Jun O

Rapaprotin is Activated by an Endopeptidase to Disassemble 26S Proteasome

雷帕蛋白酶被内肽酶激活,从而解离26S蛋白酶体。

Peng, Hanjing; Guo, Zufeng; Wang, Wei Li; Yin, Deyao; Zou, Shitao; Asbell, Thomas; Ullman, Brett R; Thakar, Maya; Zhang, Feiran; Hong, Sam Y; Rao, A V Subba; Wang, Kunyu; Zhang, Shuwen; Wu, Zhaolong; Li, Xuemei; Margolis, Seth S; Matsui, William H; Gocke, Christian B; Mao, Youdong; Liu, Jun O

Design and Synthesis of Tetrazole- and Pyridine-Containing Itraconazole Analogs as Potent Angiogenesis Inhibitors

设计并合成含四唑和吡啶的伊曲康唑类似物作为强效血管生成抑制剂

Li, Yingjun; Pasunooti, Kalyan Kumar; Peng, Hanjing; Li, Ruo-Jing; Shi, Wei Q; Liu, Wukun; Cheng, Zhiqiang; Head, Sarah A; Liu, Jun O

Rapamycin-inspired macrocycles with new target specificity

雷帕霉素启发的具有新型靶向特异性的大环化合物

Guo, Zufeng; Hong, Sam Y; Wang, Jingxin; Rehan, Shahid; Liu, Wukun; Peng, Hanjing; Das, Manisha; Li, Wei; Bhat, Shridhar; Peiffer, Brandon; Ullman, Brett R; Tse, Chung-Ming; Tarmakova, Zlatina; Schiene-Fischer, Cordelia; Fischer, Gunter; Coe, Imogen; Paavilainen, Ville O; Sun, Zhaoli; Liu, Jun O

Discovery of a Potent GLUT Inhibitor from a Library of Rapafucins by Using 3D Microarrays

利用三维微阵列技术从雷帕霉素库中发现强效GLUT抑制剂

Guo, Zufeng; Cheng, Zhiqiang; Wang, Jingxin; Liu, Wukun; Peng, Hanjing; Wang, Yuefan; Rao, A V Subba; Li, Ruo-Jing; Ying, Xue; Korangath, Preethi; Liberti, Maria V; Li, Yingjun; Xie, Yongmei; Hong, Sam Y; Schiene-Fischer, Cordelia; Fischer, Gunter; Locasale, Jason W; Sukumar, Saraswati; Zhu, Heng; Liu, Jun O

Activation of BMP Signaling by FKBP12 Ligands Synergizes with Inhibition of CXCR4 to Accelerate Wound Healing.

FKBP12 配体激活 BMP 信号通路与抑制 CXCR4 协同作用,加速伤口愈合

Peiffer Brandon J, Qi Le, Ahmadi Ali R, Wang Yuefan, Guo Zufeng, Peng Hanjing, Sun Zhaoli, Liu Jun O

An unexpected copper catalyzed 'reduction' of an arylazide to amine through the formation of a nitrene intermediate

出乎意料的是,铜催化芳基叠氮化物通过形成氮烯中间体而“还原”为胺。

Peng, Hanjing; Dornevil, Kednerlin H; Draganov, Alexander B; Chen, Weixuan; Dai, Chaofeng; Nelson, William H; Liu, Aimin; Wang, Binghe

Thiol reactive probes and chemosensors

硫醇反应探针和化学传感器

Peng, Hanjing; Chen, Weixuan; Cheng, Yunfeng; Hakuna, Lovemore; Strongin, Robert; Wang, Binghe

A fluorescent probe for fast and quantitative detection of hydrogen sulfide in blood

一种用于快速定量检测血液中硫化氢的荧光探针

Peng, Hanjing; Cheng, Yunfeng; Dai, Chaofeng; King, Adrienne L; Predmore, Benjamin L; Lefer, David J; Wang, Binghe