Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms
发现一种高选择性JAK2抑制剂BMS-911543,用于治疗骨髓增生性肿瘤
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5b00226
Wan, Honghe; Schroeder, Gretchen M; Hart, Amy C; Inghrim, Jennifer; Grebinski, James; Tokarski, John S; Lorenzi, Matthew V; You, Dan; Mcdevitt, Theresa; Penhallow, Becky; Vuppugalla, Ragini; Zhang, Yueping; Gu, Xiaomei; Iyer, Ramaswamy; Lombardo, Louis J; Trainor, George L; Ruepp, Stefan; Lippy, Jonathan; Blat, Yuval; Sack, John S; Khan, Javed A; Stefanski, Kevin; Sleczka, Bogdan; Mathur, Arvind; Sun, Jung-Hui; Wong, Michael K; Wu, Dauh-Rurng; Li, Peng; Gupta, Anuradha; Arunachalam, P N; Pragalathan, Bala; Narayanan, Sankara; K C, Nanjundaswamy; Kuppusamy, Prakasam; Purandare, Ashok V