日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Upregulation of ALDH1 as an adaptive epigenetic response to anthracyclines in acute myeloid leukemia

ALDH1上调是急性髓系白血病中蒽环类药物的一种适应性表观遗传反应。

Francesco Leonetti ,Sladjana Kosanovic ,Rocio Rebollidos-Rios ,Iris Manosalva ,Céline Baier ,Muhube Yazir ,Andrada Constantinescu ,Charbel Souaid ,Raquel Pequerul ,Miroslava Kari Adamcova ,Mehak Shaikh ,Magdalena Havlová ,Regis Costello ,Jaume Farrés ,Guillaume Martin ,Meritxell Alberich-Jorda ,Salvatore Spicuglia ,Mileidys Perez-Alea

Discovery of a reversible ALDH1A3 inhibitor throwugh a consensus docking-based virtual screening study

通过基于共识对接的虚拟筛选研究发现了一种可逆的ALDH1A3抑制剂

Batlle, E; Pequerul, R; Farrés, J; Eriksson, L A; Pors, K; Jha, V

Targeting Retinaldehyde Dehydrogenases to Enhance Temozolomide Therapy in Glioblastoma.

靶向视黄醛脱氢酶以增强替莫唑胺治疗胶质母细胞瘤的效果

Jiménez Rafael, Constantinescu Andrada, Yazir Muhube, Alfonso-Triguero Paula, Pequerul Raquel, Parés Xavier, Pérez-Alea Mileidys, Candiota Ana Paula, Farrés Jaume, Lorenzo Julia

Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer

4-(二乙氨基)苯甲醛支架的扩展探讨其对前列腺癌醛脱氢酶活性和抗增殖活性的影响

Ali I M Ibrahim, Elisabet Batlle, Smarakan Sneha, Rafael Jiménez, Raquel Pequerul, Xavier Parés, Till Rüngeler, Vibhu Jha, Tiziano Tuccinardi, Maria Sadiq, Fiona Frame, Norman J Maitland, Jaume Farrés, Klaus Pors

Structural and biochemical evidence that ATP inhibits the cancer biomarker human aldehyde dehydrogenase 1A3

结构和生化证据表明,ATP抑制癌症生物标志物人醛脱氢酶1A3

Castellví, Albert; Pequerul, Raquel; Barracco, Vito; Juanhuix, Judith; Parés, Xavier; Farrés, Jaume