日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulfilimines: An Underexplored Bioisostere for Drug Design?

亚磺酰亚胺:药物设计中尚未充分开发的生物等排体?

Arvidsson, Per I

Development and in vitro evaluation of 1,4,7-triazacyclononane-coupled β-lactams against metallo-β-lactamase producing bacteria

1,4,7-三氮杂环壬烷偶联β-内酰胺类抗生素对产金属β-内酰胺酶细菌的体外开发和评价

Shungube, Mbongeni; Reddy, Nakita; Ghazi, Terisha; Govender, Kimberleigh B; Singh, Ravesh; Kajee, Afsana; Chuturgoon, Anil; Kruger, Hendrik G; Arvidsson, Per I; Tiwari, Dileep; Govender, Thavendran; Naicker, Tricia

Base-Mediated Tandem Michael Addition and SuFEx Cyclization for the Synthesis of Sultone-Containing Spirooxindoles

碱催化串联迈克尔加成和SuFEx环化反应合成含磺内酯的螺环氧吲哚

Govender, Kimberleigh B; Simelane, Sandile B; Chetty, Lloyd C; Kruger, Hendrik G; Govender, Thavendran; Arvidsson, Per I; Naicker, Tricia

Navigating the complexities of drug development for metallo-β-lactamase inhibitors

应对金属β-内酰胺酶抑制剂药物研发的复杂性

Reddy, Nakita; Balieiro, Alessandra Moraes; Silva, José Rogério A; Gouws, Christiaan A; Mutshembele, Awelani; Arvidsson, Per I; Kruger, Hendrik G; Govender, Thavendran; Naicker, Tricia

Facile Synthesis of Oxazolidinones as Potential Antibacterial Agents

简便合成噁唑烷酮类化合物作为潜在抗菌剂

Els, Secret P; Govender, Kimberleigh B; Sokhela, Mxolisi K; Bhatt, Nilay; Reddy, Nakita; Kruger, Hendrik G; Arvidsson, Per I; Gunosewoyo, Hendra; Govender, Thavendran; Naicker, Tricia

Investigating the efficacy of green solvents and solvent-free conditions in hydrogen-bonding mediated organocatalyzed model reactions

研究绿色溶剂和无溶剂条件在氢键介导的有机催化模型反应中的有效性

Chetty, Lloyd C; Kruger, Hendrik G; Arvidsson, Per I; Naicker, Tricia; Govender, Thavendran

The Oxidation of Electron-Rich Arenes Using a H(2)O(2)-Proline System

利用H₂O₂-脯氨酸体系氧化富电子芳烃

Chetty, Lloyd C; Kruger, Hendrik G; Arvidsson, Per I; Maguire, Glenn E M; Govender, Thavendran; Naicker, Tricia

Neutralizing Carbapenem Resistance by Co-Administering Meropenem with Novel β-Lactam-Metallo-β-Lactamase Inhibitors

美罗培南与新型β-内酰胺-金属-β-内酰胺酶抑制剂联合用药可中和碳青霉烯耐药性

Reddy, Nakita; Girdhari, Letisha; Shungube, Mbongeni; Gouws, Arnoldus C; Peters, Byron K; Rajbongshi, Kamal K; Baijnath, Sooraj; Mdanda, Sipho; Ntombela, Thandokuhle; Arumugam, Thilona; Bester, Linda A; Singh, Sanil D; Chuturgoon, Anil; Arvidsson, Per I; Maguire, Glenn E M; Kruger, Hendrik G; Govender, Thavendran; Naicker, Tricia

In Vitro and In Vivo Development of a β-Lactam-Metallo-β-Lactamase Inhibitor: Targeting Carbapenem-Resistant Enterobacterales

β-内酰胺-金属-β-内酰胺酶抑制剂的体外和体内开发:针对耐卡巴培南类抗生素的肠杆菌

Byron K Peters, Nakita Reddy, Mbongeni Shungube, Letisha Girdhari, Sooraj Baijnath, Sipho Mdanda, Lloyd Chetty, Thandokuhle Ntombela, Thilona Arumugam, Linda A Bester, Sanil D Singh, Anil Chuturgoon, Per I Arvidsson, Glenn E M Maguire, Hendrik G Kruger, Tricia Naicker, Thavendran Govender

Shock-Induced Endothelial Dysfunction is Present in Patients With Occult Hypoperfusion After Trauma

创伤后隐匿性低灌注患者存在休克诱发的内皮功能障碍

Heather R Kregel, Gabrielle E Hatton, Kayla D Isbell, Hanne H Henriksen, Jakob Stensballe, Per I Johansson, Lillian S Kao, Charles E Wade