日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fused 3D boron heterocycles via EnT catalysis: synthesis, modification and validation as beta-lactamase inhibitors

通过 EnT 催化合成稠合三维硼杂环化合物:合成、修饰及作为 β-内酰胺酶抑制剂的验证

Kortman, Hannah M; Fang, Hao; Bastick, Kane A C; Völkel, Charlotte; Oberthür, Dominik; Seeberger, Peter H; Perbandt, Markus; Molloy, John J

Time-resolved crystallography of boric acid binding to the active site serine of the β-lactamase CTX-M-14 and subsequent 1,2-diol esterification

利用时间分辨晶体学方法研究硼酸与β-内酰胺酶CTX-M-14活性位点丝氨酸结合及其后续的1,2-二醇酯化反应。

Prester, Andreas; Perbandt, Markus; Galchenkova, Marina; Oberthuer, Dominik; Werner, Nadine; Henkel, Alessandra; Maracke, Julia; Yefanov, Oleksandr; Hakanpää, Johanna; Pompidor, Guillaume; Meyer, Jan; Chapman, Henry; Aepfelbacher, Martin; Hinrichs, Winfried; Rohde, Holger; Betzel, Christian

Antiviral activity of natural phenolic compounds in complex at an allosteric site of SARS-CoV-2 papain-like protease

天然酚类化合物与SARS-CoV-2木瓜蛋白酶样蛋白酶变构位点形成复合物的抗病毒活性

Srinivasan, Vasundara; Brognaro, Hévila; Prabhu, Prince R; de Souza, Edmarcia Elisa; Günther, Sebastian; Reinke, Patrick Y A; Lane, Thomas J; Ginn, Helen; Han, Huijong; Ewert, Wiebke; Sprenger, Janina; Koua, Faisal H M; Falke, Sven; Werner, Nadine; Andaleeb, Hina; Ullah, Najeeb; Franca, Bruno Alves; Wang, Mengying; Barra, Angélica Luana C; Perbandt, Markus; Schwinzer, Martin; Schmidt, Christina; Brings, Lea; Lorenzen, Kristina; Schubert, Robin; Machado, Rafael Rahal Guaragna; Candido, Erika Donizette; Oliveira, Danielle Bruna Leal; Durigon, Edison Luiz; Niebling, Stephan; Garcia, Angelica Struve; Yefanov, Oleksandr; Lieske, Julia; Gelisio, Luca; Domaracky, Martin; Middendorf, Philipp; Groessler, Michael; Trost, Fabian; Galchenkova, Marina; Mashhour, Aida Rahmani; Saouane, Sofiane; Hakanpää, Johanna; Wolf, Markus; Alai, Maria Garcia; Turk, Dusan; Pearson, Arwen R; Chapman, Henry N; Hinrichs, Winfried; Wrenger, Carsten; Meents, Alke; Betzel, Christian

Structural basis to repurpose boron-based proteasome inhibitors Bortezomib and Ixazomib as β-lactamase inhibitors

将硼基蛋白酶体抑制剂硼替佐米和伊沙佐米重新用作β-内酰胺酶抑制剂的结构基础

Perbandt, Markus; Werner, Nadine; Prester, Andreas; Rohde, Holger; Aepfelbacher, Martin; Hinrichs, Winfried; Betzel, Christian

Structure and activity of the DHNA Coenzyme-A Thioesterase from Staphylococcus aureus providing insights for innovative drug development

金黄色葡萄球菌DHNA辅酶A硫酯酶的结构和活性为创新药物研发提供了见解

Murad, Aline Melro; Brognaro, Hévila; Falke, Sven; Lindner, Jasmin; Perbandt, Markus; Mudogo, Celestin; Schubert, Robin; Wrenger, Carsten; Betzel, Christian

Rapid and efficient room-temperature serial synchrotron crystallography using the CFEL TapeDrive

利用CFEL TapeDrive实现快速高效的室温串行同步辐射晶体学研究

Zielinski, Kara A; Prester, Andreas; Andaleeb, Hina; Bui, Soi; Yefanov, Oleksandr; Catapano, Lucrezia; Henkel, Alessandra; Wiedorn, Max O; Lorbeer, Olga; Crosas, Eva; Meyer, Jan; Mariani, Valerio; Domaracky, Martin; White, Thomas A; Fleckenstein, Holger; Sarrou, Iosifina; Werner, Nadine; Betzel, Christian; Rohde, Holger; Aepfelbacher, Martin; Chapman, Henry N; Perbandt, Markus; Steiner, Roberto A; Oberthuer, Dominik

Crystal structure of an extracellular superoxide dismutase from Onchocerca volvulus and implications for parasite-specific drug development

盘尾丝虫胞外超氧化物歧化酶的晶体结构及其对寄生虫特异性药物研发的意义

Moustafa, Amr; Perbandt, Markus; Liebau, Eva; Betzel, Christian; Falke, Sven

The Komagataeibacter europaeus GqqA is the prototype of a novel bifunctional N-Acyl-homoserine lactone acylase with prephenate dehydratase activity

Komagataeibacter europaeus GqqA 是一种新型双功能 N-酰基高丝氨酸内酯酰化酶的原型,具有预苯酸脱水酶活性

Nadine Werner #, Katrin Petersen #, Christel Vollstedt, Pablo Perez Garcia, Jennifer Chow, Manuel Ferrer, Laura Fernandez-Lopez, Sven Falke, Markus Perbandt, Winfried Hinrichs, Christian Betzel, Wolfgang R Streit

In cellulo crystallization of Trypanosoma brucei IMP dehydrogenase enables the identification of genuine co-factors

布氏锥虫 IMP 脱氢酶的纤维素结晶能够识别真正的辅助因子

Karol Nass #, Lars Redecke #, M Perbandt, O Yefanov, M Klinge, R Koopmann, F Stellato, A Gabdulkhakov, R Schönherr, D Rehders, J M Lahey-Rudolph, A Aquila, A Barty, S Basu, R B Doak, R Duden, M Frank, R Fromme, S Kassemeyer, G Katona, R Kirian, H Liu, I Majoul, J M Martin-Garcia, M Messerschmidt, R

A Giant Extracellular Matrix Binding Protein of Staphylococcus epidermidis Binds Surface-Immobilized Fibronectin via a Novel Mechanism

表皮葡萄球菌的巨大细胞外基质结合蛋白通过新机制与表面固定的纤连蛋白结合

Henning Büttner, Markus Perbandt, Thomas Kohler, Alexey Kikhney, Manuel Wolters, Martin Christner, Marisol Heise, Jérôme Wilde, Samira Weißelberg, Anna Both, Christian Betzel, Sven Hammerschmidt, Dmitri Svergun, Martin Aepfelbacher, Holger Rohde