日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

BMS-986251 的发现:一种临床上可行、高效且选择性的 RORγt 反向激动剂

Cherney, Robert J; Cornelius, Lyndon A M; Srivastava, Anurag; Weigelt, Carolyn A; Marcoux, David; Duan, James J-W; Shi, Qing; Batt, Douglas G; Liu, Qingjie; Yip, Shiuhang; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John; Khan, Javed; Wang, Jinhong; Yarde, Melissa; Cvijic, Mary Ellen; Mathur, Arvind; Li, Sha; Shuster, David; Khandelwal, Purnima; Borowski, Virna; Xie, Jenny; Obermeier, Mary; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Tino, Joseph A; Macor, John E; Salter-Cid, Luisa; Denton, Rex; Zhao, Qihong; Carter, Percy H; Dhar, T G Murali

Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK

利用旋转稳定的阻转异构体增强效力:发现吡啶并嘧啶二酮-咔唑类BTK抑制剂

Srivastava, Anurag S; Ko, Soo; Watterson, Scott H; Pattoli, Mark A; Skala, Stacey; Cheng, Lihong; Obermeier, Mary T; Vickery, Rodney; Discenza, Lorell N; D'Arienzo, Celia J; Gillooly, Kathleen M; Taylor, Tracy L; Pulicicchio, Claudine; McIntyre, Kim W; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Dai, Jun; Wang, Chunlei; Zhang, Yingru; Wang, Bei; Pawluczyk, Joseph; Kempson, James; Zhao, Rulin; Hou, Xiaoping; Rampulla, Richard; Mathur, Arvind; Galella, Michael A; Salter-Cid, Luisa; Barrish, Joel C; Carter, Percy H; Fura, Aberra; Burke, James R; Tino, Joseph A

Aryl Ether-Derived Sphingosine-1-Phosphate Receptor (S1P(1)) Modulators: Optimization of the PK, PD, and Safety Profiles

芳基醚衍生的鞘氨醇-1-磷酸受体(S1P(1))调节剂:药代动力学、药效学和安全性特征的优化

Xiao, Zili; Yang, Michael G; Dhar, T G Murali; Xiao, Hai-Yun; Gilmore, John L; Marcoux, David; McIntyre, Kim W; Taylor, Tracy L; Shi, Hong; Levesque, Paul C; Marino, Anthony M; Cornelius, Georgia; Mathur, Arvind; Shen, Ding Ren; Cvijic, Mary Ellen; Lehman-McKeeman, Lois D; Sun, Huadong; Xie, Jenny H; Carter, Percy H; Dyckman, Alaric J

Identification of potent tricyclic prodrug S1P(1) receptor modulators

鉴定强效三环类前药S1P(1)受体调节剂

Marcoux, David; Xiao, Hai-Yun; Murali Dhar, T G; Xie, Jenny; Lehman-McKeeman, Lois D; Wu, Dauh-Rurng; Dabros, Marta; Yang, Xiaoxia; Taylor, Tracy L; Zhou, Xia D; Heimrich, Elizabeth M; Thomas, Rochelle; McIntyre, Kim W; Shi, Hong; Levesque, Paul C; Sun, Huadong; Yang, Zheng; Marino, Anthony M; Cornelius, Georgia; D'Arienzo, Celia J; Gupta, Anuradha; Pragalathan, Bala; Rampulla, Richard; Mathur, Arvind; Shen, Ding Ren; Cvijic, Mary Ellen; Salter-Cid, Luisa; Lombardo, Louis J; Carter, Percy H; Dyckman, Alaric J

Investigating investment in biopharmaceutical R&D

调查对生物制药研发的投资

Carter, Percy H; Berndt, Ernst R; DiMasi, Joseph A; Trusheim, Mark

Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials

BMS-986104的鉴定和临床前药理学研究:一种在临床试验中应用的差异化S1P1受体调节剂

Dhar, T G Murali; Xiao, Hai-Yun; Xie, Jenny; Lehman-McKeeman, Lois D; Wu, Dauh-Rurng; Dabros, Marta; Yang, Xiaoxia; Taylor, Tracy L; Zhou, Xia D; Heimrich, Elizabeth M; Thomas, Rochelle; McIntyre, Kim W; Warrack, Bethanne; Shi, Hong; Levesque, Paul C; Zhu, Jia L; Hennan, James; Balimane, Praveen; Yang, Zheng; Marino, Anthony M; Cornelius, Georgia; D'Arienzo, Celia J; Mathur, Arvind; Shen, Ding Ren; Cvijic, Mary Ellen; Salter-Cid, Luisa; Barrish, Joel C; Carter, Percy H; Dyckman, Alaric J

Alkylsulfone-containing trisubstituted cyclohexanes as potent and bioavailable chemokine receptor 2 (CCR2) antagonists

含烷基砜的三取代环己烷作为强效且生物利用度高的趋化因子受体2 (CCR2) 拮抗剂

Cherney, Robert J; Mo, Ruowei; Yang, Michael G; Xiao, Zili; Zhao, Qihong; Mandlekar, Sandhya; Cvijic, Mary Ellen; Charo, Israel F; Barrish, Joel C; Decicco, Carl P; Carter, Percy H

Discovery of disubstituted cyclohexanes as a new class of CC chemokine receptor 2 antagonists

发现双取代环己烷作为一类新型 CC 趋化因子受体 2 拮抗剂

Robert J Cherney, Ruowei Mo, Dayton T Meyer, David J Nelson, Yvonne C Lo, Gengjie Yang, Peggy A Scherle, Sandhya Mandlekar, Zelda R Wasserman, Heather Jezak, Kimberly A Solomon, Andrew J Tebben, Percy H Carter, Carl P Decicco

An apparatus for delivery of electroconvulsive shock without situational change

一种无需改变环境即可施加电休克的装置。

Grosser, G S; Percy, H E