日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pleiotropic prodrugs for both symptomatic and disease-modifying treatment of Alzheimer's disease

用于治疗阿尔茨海默病症状和改善疾病进程的多效性前药

Meden, Anže; Žnidaršič, Neža; Knez, Damijan; Wang, Yuanyuan; Xu, Ziwei; Yang, Huajing; Zhang, Weiting; Pišlar, Anja; Perdih, Andrej; Brezar, Simona Kranjc; Grgurevič, Neža; Pajk, Stane; Sun, Haopeng; Gobec, Stanislav

Access to amidines via C(sp(2))-N coupling of trifluoroborate-iminiums with N-fluorobenzenesulfonimide

通过三氟硼酸亚胺与N-氟苯磺酰亚胺的C(sp(2))-N偶联反应合成脒类化合物

Knez, Damijan; Šterman, Andrej; Sosič, Izidor; Perdih, Franc; Nuñez, Gonzalo D; Knaflič, Tilen; Arčon, Denis; Besora, Maria; Carbó, Jorge J; Fernández, Elena; Časar, Zdenko

Water-Based Pharmacophore Modeling in Kinase Inhibitor Design: A Case Study on Fyn and Lyn Protein Kinases

水基药效团模型在激酶抑制剂设计中的应用:以Fyn和Lyn蛋白激酶为例

Ljubič, Martin; Sollner Dolenc, Marija; Borišek, Jure; Perdih, Andrej

Influenza a Virus Inhibition: Evaluating Computationally Identified Cyproheptadine Through In Vitro Assessment

甲型流感病毒抑制:通过体外评估评价计算机筛选出的赛庚啶

Glisic, Sanja; Stevanovic, Kristina; Perdih, Andrej; Bukreyeva, Natalya; Maruyama, Junki; Perovic, Vladimir; López-Serrano, Sergi; Darji, Ayub; Radosevic, Draginja; Sencanski, Milan; Veljkovic, Veljko; Botta, Bruno; Mori, Mattia; Paessler, Slobodan

Mediators of outcome in adolescent psychotherapy and their implications for theories and mechanisms of change: a systematic review

青少年心理治疗结果的中介因素及其对理论和改变机制的启示:一项系统性综述

Taubner, Svenja; Ioannou, Yianna; Saliba, Andrea; Sales, Célia M D; Volkert, Jana; Protić, Sonja; Adler, Asta; Barkauskiene, Rasa; Conejo-Cerón, Sonia; Di Giacomo, Dina; Mestre, Jose M; Moreno-Peral, Patricia; Vieira, Filipa Mucha; Mota, Catarina Pinheiro; Henriques, Margarida Isabel Rangel Santos; Røssberg, Jan Ivar; Perdih, Tjasa Stepisnik; Schmidt, Stefanie Julia; Zettl, Max; Ulberg, Randi; Heinonen, Erkki

2-Bromopyridines as Versatile Synthons for Heteroarylated 2-Pyridones via Ru(II)-Mediated Domino C-O/C-N/C-C Bond Formation Reactions

2-溴吡啶作为多功能合成子,通过Ru(II)介导的多米诺CO/CN/CC键形成反应合成杂芳基化2-吡啶酮

Drev, Miha; Brodnik, Helena; Grošelj, Uroš; Perdih, Franc; Svete, Jurij; Štefane, Bogdan; Požgan, Franc

Simulation- and AI-directed optimization of 4,6-substituted 1,3,5-triazin-2(1 H)-ones as inhibitors of human DNA topoisomerase IIα

模拟和人工智能指导优化 4,6-取代的 1,3,5-三嗪-2(1H)-酮作为人类 DNA 拓扑异构酶 IIα 抑制剂

Barbara Herlah, Tjaša Goričan, Nika Strašek Benedik, Simona Golič Grdadolnik, Izidor Sosič, Andrej Perdih

Expanding the Structural Diversity at the Phenylene Core of Ligands for the von Hippel-Lindau E3 Ubiquitin Ligase: Development of Highly Potent Hypoxia-Inducible Factor-1α Stabilizers

扩大 von Hippel-Lindau E3 泛素连接酶配体苯基核心的结构多样性:开发高效缺氧诱导因子-1α 稳定剂

Lan Phuong Vu, Claudia J Diehl, Ryan Casement, Adam G Bond, Christian Steinebach, Nika Strašek, Aleša Bricelj, Andrej Perdih, Gregor Schnakenburg, Izidor Sosič, Alessio Ciulli, Michael Gütschow

Three-Component Reaction of 3-Formyl-6-Methylchromone, Primary Amines, and Secondary Phosphine Oxides: A Synthetic and Mechanistic Study

3-甲酰基-6-甲基色酮、伯胺和仲膦氧化物的三组分反应:合成与机理研究

Popovics-Tóth, Nóra; Bao, Trinh Dang Tran; Tajti, Ádám; Mátravölgyi, Béla; Kelemen, Zsolt; Perdih, Franc; Hackler, László Jr; Puskás, László G; Bálint, Erika

Unveiling the interdomain dynamics of type II DNA topoisomerase through all-atom simulations: Implications for understanding its catalytic cycle

通过全原子模拟揭示II型DNA拓扑异构酶的结构域间动力学:对理解其催化循环的启示

Pavlin, Matic; Herlah, Barbara; Valjavec, Katja; Perdih, Andrej