日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proximity-Induced Rewiring of Oncogenic Kinase Triggers Apoptosis

邻近诱导的致癌激酶重编程触发细胞凋亡

Merz, Manuel L; Shoba, Veronika M; Pergu, Rajaiah; Severance, Zachary C; Munkanatta Godage, Dhanushka N P; Deb, Arghya; Kwok, Hui Si; Singh, Prashant; Singh, Sameek; Allen, Jonathan B; Tian, Wenzhi; Gosavi, Pallavi M; Chaudhary, Santosh K; Anokhina, Viktoriya; Weisberg, Ellen L; Payne, N Connor; He, Yao; Dhaliwal, Rohil; Osadchey, Reilly; Shekhar, Mrinal; Mazitschek, Ralph; Rees, Matthew G; Roth, Jennifer A; Cui, Qiang; Griffin, James D; Liau, Brian B; Choudhary, Amit

A Scalable Design for Proximity-Inducing Molecules

一种可扩展的邻近诱导分子设计

Karaj, Endri; Venkatarangan, Varsha; Sindi, Shaimaa H; Siriwongsup, Surached; Lee, Chaiheon; Pergu, Rajaiah; Sreekanth, Vedagopuram; Kailass, Karishma; Tran, Kien; Singh, Prashant; Singh, Sameek; Kawai, Junya; Fung, Jeffrey E; Tefera, Mahilet; Dhaliwal, Rohil; Chaudhary, Santosh K; Keyes, April; Sadagopan, Ananthan; Boatner, Lisa; Shah, Neel H; Fehl, Charlie; Backus, Keriann M; Choudhary, Amit

Phosphorylation-Inducing Molecules for Regulating Dynamic Cellular Processes

调控动态细胞过程的磷酸化诱导分子

Pergu, Rajaiah; Sreekanth, Vedagopuram; Kokkonda, Praveen; Lai, Sophia; Tiwari, Praveen K; Singh, Sameek; Kawai, Junya; Singha, Santanu; Tian, Wenzhi; Thimaradka, Vikram; Siriwongsup, Surached; Tran, Kien; Choudhary, Amit

Ultrasmall chemogenetic tags with group-transfer ligands

带有基团转移配体的超小型化学遗传标签

Vedagopuram, Sreekanth; Sindi, Shaimaa; Chaudhary, Santosh K; Pergu, Rajaiah; Singh, Prashant; Karaj, Endri; Fung, Jeffrey E; Deb, Arghya; DeCarlo, Stephan J; Mercer, Jaron A M; Yamada, Kei; Rodriguez, Diego; Liu, David R; Choudhary, Amit

Orthogonal resistance mechanisms of classical- and induced-proximity inhibitors.

经典邻近抑制剂和诱导邻近抑制剂的正交耐药机制

Merz Manuel L, Kailass Karishma, Pergu Rajaiah, Tran Kien, Gupta Kritika, Severance Zachary C, Singh Sameek, Vedagopuram Sreekanth, Law Benjamin K, Rosenblatt Gideon, Dhaliwal Rohil, Choudhary Amit

Phosphorylation-inducing chimera rewires oncogenic kinase to trigger apoptosis.

磷酸化诱导嵌合体重塑致癌激酶以触发细胞凋亡

Merz Manuel L, Shoba Veronika M, Pergu Rajaiah, Severance Zachary C, Munkanatta Godage Dhanushka N P, Deb Arghya, Kwok Hui Si, Singh Prashant, Singh Sameek, Allen Jonathan B, Tian Wenzhi, Gosavi Pallavi M, Chaudhary Santosh K, Anokhina Viktoriya, Weisberg Ellen L, Payne N Connor, He Yao, Osadchey Reilly, Shekhar Mrinal, Mazitschek Ralph, Rees Matthew G, Roth Jennifer A, Cui Qiang, Griffin James D, Liau Brian B, Choudhary Amit

Development and Applications of Chimera Platforms for Tyrosine Phosphorylation

酪氨酸磷酸化嵌合平台的开发与应用

Pergu, Rajaiah; Shoba, Veronika M; Chaudhary, Santosh K; Munkanatta Godage, Dhanushka N P; Deb, Arghya; Singha, Santanu; Dhawa, Uttam; Singh, Prashant; Anokhina, Viktoriya; Singh, Sameek; Siriwardena, Sachini U; Choudhary, Amit

A general approach to identify cell-permeable and synthetic anti-CRISPR small molecules

识别可穿透细胞且合成的抗 CRISPR 小分子的通用方法

Donghyun Lim #, Qingxuan Zhou #, Kurt J Cox #, Benjamin K Law #, Miseon Lee #, Praveen Kokkonda #, Vedagopuram Sreekanth #, Rajaiah Pergu, Santosh K Chaudhary, Soumyashree A Gangopadhyay, Basudeb Maji, Sophia Lai, Yuka Amako, David B Thompson, Hari K K Subramanian, Michael F Mesleh, Vlado Dančík, Pa

Phosphorylation and Pin1 binding to the LIC1 subunit selectively regulate mitotic dynein functions

磷酸化和 Pin1 与 LIC1 亚基的结合选择性地调节有丝分裂动力蛋白的功能

Amrita Kumari, Chandan Kumar, Rajaiah Pergu, Megha Kumar, Sagar P Mahale, Neeraj Wasnik, Sivaram V S Mylavarapu

Chemogenetic System Demonstrates That Cas9 Longevity Impacts Genome Editing Outcomes

化学遗传系统证明 Cas9 寿命影响基因组编辑结果

Vedagopuram Sreekanth, Qingxuan Zhou, Praveen Kokkonda, Heysol C Bermudez-Cabrera, Donghyun Lim, Benjamin K Law, Benjamin R Holmes, Santosh K Chaudhary, Rajaiah Pergu, Brittany S Leger, James A Walker, David K Gifford, Richard I Sherwood, Amit Choudhary