日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and structure-activity relationship studies of small molecule disruptors of EWS-FLI1 interactions in Ewing's sarcoma

尤文氏肉瘤中 EWS-FLI1 相互作用的小分子干扰物的合成及构效关系研究

Perrer N Tosso, Yali Kong, Lauren Scher, Ryan Cummins, Jeffrey Schneider, Said Rahim, K Travis Holman, Jeffrey Toretsky, Kan Wang, Aykut Üren, Milton L Brown

Single enantiomer of YK-4-279 demonstrates specificity in targeting the oncogene EWS-FLI1

YK-4-279 的单一对映异构体对靶向癌基因 EWS-FLI1 表现出特异性。

Barber-Rotenberg, Julie S; Selvanathan, Saravana P; Kong, Yali; Erkizan, Hayriye V; Snyder, Tara M; Hong, S Peter; Kobs, Christina L; South, Natalie L; Summer, Steven; Monroe, Philip J; Chruszcz, Maksymilian; Dobrev, Veselin; Tosso, Perrer N; Scher, Lauren J; Minor, Wladek; Brown, Milton L; Metallo, Steven J; Üren, Aykut; Toretsky, Jeffrey A