Discovery of GSK8612, a Highly Selective and Potent TBK1 Inhibitor
发现高选择性和强效的TBK1抑制剂GSK8612
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.9b00027
Thomson, Douglas W; Poeckel, Daniel; Zinn, Nico; Rau, Christina; Strohmer, Katrin; Wagner, Anne J; Graves, Alan P; Perrin, Jessica; Bantscheff, Marcus; Duempelfeld, Birgit; Kasparcova, Viera; Ramanjulu, Joshi M; Pesiridis, G Scott; Muelbaier, Marcel; Bergamini, Giovanna