Discovery of 1H-pyrazol-3(2H)-ones as potent and selective inhibitors of protein kinase R-like endoplasmic reticulum kinase (PERK)
发现 1H-吡唑-3(2H)-酮是蛋白激酶 R 样内质网激酶 (PERK) 的有效和选择性抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm5017494
Adrian L Smith, Kristin L Andrews, Holger Beckmann, Steven F Bellon, Pedro J Beltran, Shon Booker, Hao Chen, Young-Ah Chung, Noel D D'Angelo, Jennifer Dao, Kenneth R Dellamaggiore, Peter Jaeckel, Richard Kendall, Katja Labitzke, Alexander M Long, Silvia Materna-Reichelt, Petia Mitchell, Mark H Norma
