Conversion of Bim-BH3 from Activator to Inhibitor of Bak through Structure-Based Design
通过基于结构的设计将 Bim-BH3 从 Bak 激活剂转化为抑制剂
期刊:Molecular Cell
影响因子:14.5
doi:10.1016/j.molcel.2017.11.001
Jason M Brouwer, Ping Lan, Angus D Cowan, Jonathan P Bernardini, Richard W Birkinshaw, Mark F van Delft, Brad E Sleebs, Adeline Y Robin, Ahmad Wardak, Iris K Tan, Boris Reljic, Erinna F Lee, W Douglas Fairlie, Melissa J Call, Brian J Smith, Grant Dewson, Guillaume Lessene, Peter M Colman, Peter E Cz