日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A novel long-acting relaxin-2 fusion, AZD3427, improves cardiac performance in non-human primates with cardiac dysfunction.

一种新型长效松弛素-2融合蛋白AZD3427可改善患有心脏功能障碍的非人灵长类动物的心脏功能

Papworth Monika, Kulkarni Spoorthy, Antonsson Madeleine, Sermadiras Isabelle, Hovdal Daniel, Connolly Kathleen, Olsson Jan, Shukla Animesh, Cotton Peter, Althage Magnus, Paterson Judy, Martin Esther, Wolny Marcin, Ferraro Franco, Sadowska Agnieszka, Hao Weidong, Larsson Niklas, Backmark Anna, Marlow Tom, Perez Rosario, Jermutus Lutz, Omar Sami, George Richard T, Gabrielsen Anders, Pettersen Daniel, Jennbacken Karin

Re-PERFUSE: Phase 1b study of AZD3427, a novel relaxin receptor agonist, on renal perfusion in HFrEF patients

Re-PERFUSE:AZD3427(一种新型松弛素受体激动剂)对射血分数降低型心力衰竭(HFrEF)患者肾脏灌注的1b期研究

Ufnal, Marcin; Quintana-Hayashi, Macarena P; Connolly, Kathleen; Pettersen, Daniel; Cselényi, Zsolt; Jucaite, Aurelija; Schou, Magnus; Varrone, Andrea; Chan, Melanie; Lund, Lars H

Novel Relaxin Receptor RXFP1 Agonist AZD3427 in the Treatment of Heart Failure: A Phase 1a/b, First-in-Human, Randomized, Single-Blind, Placebo-Controlled Study

新型松弛素受体RXFP1激动剂AZD3427治疗心力衰竭:一项1a/b期、首次人体试验、随机、单盲、安慰剂对照研究

Connolly, Kathleen; George, Richard; Omar, Sami; Matsson, Elin; Åstrand, Magnus; Althage, Magnus; Pettersen, Daniel; Mohamed, Esha; Fang, Kelly; Lima, Joao A C; Kujacic, Mirjana; Ödesjö, Helena; Turton, Michelle; Johannesson, Petra; Gabrielsen, Anders; Ufnal, Marcin

Design of Selective sPLA(2)-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

选择性 sPLA(2)-X 抑制剂 (-)-2-{2-[氨基甲酰基-6-(三氟甲氧基)-1H-吲哚-1-基]吡啶-2-基}丙酸的设计

Giordanetto, Fabrizio; Knerr, Laurent; Nordberg, Peter; Pettersen, Daniel; Selmi, Nidhal; Beisel, Hans-Georg; de la Motte, Hannah; Månsson, Åsa; Dahlström, Mikael; Broddefalk, Johan; Saarinen, Gabrielle; Klingegård, Fredrik; Hurt-Camejo, Eva; Rosengren, Birgitta; Wikström, Johannes; Wågberg, Maria; Brengdahl, Johan; Rohman, Mattias; Sandmark, Jenny; Åkerud, Tomas; Roth, Robert G; Jansen, Frank; Ahlqvist, Marie

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie