日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

From DNA-Encoded Library Screening to AM-9747: An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo Efficacy.

从 DNA 编码文库筛选到 AM-9747:一种具有强效口服体内疗效的 MTA 协同 PRMT5 抑制剂

Sarvary Ian, Vestergaard Mikkel, Moretti Loris, Andersson Jan, Peiró Cadahía Jorge, Cowland Sanne, Flagstad Thomas, Franch Thomas, Gouliaev Alex, Husemoen Gitte, Jacso Tomas, Kronborg Titi, Kuropatnicka Aleksandra, Nadali Anna, Madsen Mads, Nielsen So Ren, Pii David, Ryborg So Ren, Soede Camillia, Allen Jennifer R, Bourbeau Matthew, Li Kexue, Liu Qingyian, Lo Mei-Chu, Madoux Franck, Mardirossian Narbe, Moriguchi Jodi, Ngo Rachel, Peng Chi-Chi, Pettus Liping, Tamayo Nuria, Wang Paul, Kapoor Rajiv, Belmontes Brian, Caenepeel Sean, Hughes Paul, Liu Siyuan, Slemmons Katherine K, Yang Yajing, Xie Fang, Ghimire-Rijal Sudipa, Mukund Susmith, Glad Sanne

Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors

氧代吡啶并[2,3-d]嘧啶类化合物作为共价L858R/T790M突变选择性表皮生长因子受体(EGFR)抑制剂

Wurz, Ryan P; Pettus, Liping H; Ashton, Kate; Brown, James; Chen, Jian Jeffrey; Herberich, Brad; Hong, Fang-Tsao; Hu-Harrington, Essa; Nguyen, Tom; St Jean, David J Jr; Tadesse, Seifu; Bauer, David; Kubryk, Michele; Zhan, Jinghui; Cooke, Keegan; Mitchell, Petia; Andrews, Kristin L; Hsieh, Faye; Hickman, Dean; Kalyanaraman, Nataraj; Wu, Tian; Reid, Darren L; Lobenhofer, Edward K; Andrews, Dina A; Everds, Nancy; Guzman, Roberto; Parsons, Andrew T; Hedley, Simon J; Tedrow, Jason; Thiel, Oliver R; Potter, Matthew; Radinsky, Robert; Beltran, Pedro J; Tasker, Andrew S