日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Fragment-Based Inhibitors of SARS-CoV-2 PL(Pro)

SARS-CoV-2 PL(Pro)片段抑制剂的发现

Wei, Qiangqiang; Taylor, Ashley J; Barmade, Mahesh Angadrao; Teuscher, Kevin B; Chowdhury, Somanath; Apakama, Chideraa; Anderson-Daniels, Jordan; Yongqing, Zhu; Schultz, David C; Rietz, Tyson A; South, Taylor M; Crow, Mackenzie M; Zhao, Bin; Amporndanai, Kangsa; Sensintaffar, John L; Phan, Jason; Cherry, Sara; Denison, Mark; Lee, Taekyu; Fesik, Stephen W

Discovery of Spiro[chromane-2,4'-piperidine] Derivatives as Irreversible Inhibitors of SARS-CoV-2 Papain-like Protease

发现螺[色满-2,4'-哌啶]衍生物作为SARS-CoV-2木瓜蛋白酶样蛋白酶的不可逆抑制剂

Wei, Qiangqiang; Taylor, Ashley J; Miriyala, Nagaraju; Barmade, Mahesh A; Gentry, Zachary O; Anderson-Daniels, Jordan; Teuscher, Kevin B; Crow, Mackenzie M; Apakama, Chideraa; South, Taylor M; Rietz, Tyson A; Amporndanai, Kangsa; Phan, Jason; Sensintaffar, John L; Denison, Mark; Lee, Taekyu; Fesik, Stephen W

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

Discovery of Small Molecules that Bind to Son of Sevenless 2 (SOS2)

发现与SOS2结合的小分子

Krzysztof M Zak, Alex G Waterson, Leonhard Geist, Nina Braun, Katja Hauer, Klaus Rumpel, Juergen Ramharter, Heinz Stadtmueller, Bernhard Wolkerstorfer, David Schoenbauer, Jianwen Cui, Jason Phan, Jason R Abbott, Dhruba Sarkar, Timothy R Hodges, Allison Arnold, John L Sensintaffar, Stephen W Fesik, D

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W

Nuclear Magnetic Resonance-based fragment screen of the E3 ligase Fem-1 homolog B

基于核磁共振的E3连接酶Fem-1同源物B片段筛选

Katinas, Jade M; Amporndanai, Kangsa; Taylor, Ashley J; Rose, Kristie L; Gareiss, Peter C; Crespo, Roberto A; Phan, Jason; Waterson, Alex G; Fesik, Stephen W

Identification of ligands for E3 ligases with restricted expression using fragment-based methods

利用基于片段的方法鉴定表达受限的E3连接酶的配体

Waterson, Alex G; Lehmann, Brian D; Lu, Zhenwei; Sensintaffar, John L; Olejniczak, Edward T; Zhao, Bin; Rietz, Tyson; Payne, William G; Phan, Jason; Fesik, Stephen W

Fragment-Based Screen of SARS-CoV-2 Papain-like Protease (PL(pro))

基于片段的SARS-CoV-2木瓜蛋白酶样蛋白酶(PL(pro))筛选

Taylor, Ashley J; Amporndanai, Kangsa; Rietz, Tyson A; Zhao, Bin; Thiruvaipati, Anusha; Wei, Qiangqiang; South, Taylor M; Crow, Mackenzie M; Apakama, Chideraa; Sensintaffar, John L; Phan, Jason; Lee, Taekyu; Fesik, Stephen W

Confinement plus myosin-II suppression maximizes heritable loss of chromosomes, as revealed by live-cell ChReporters

活细胞 ChReporters 研究表明,限制细胞活动并抑制肌球蛋白 II 可最大程度地导致遗传性染色体丢失。

Brandon H Hayes ,Peter Kuangzheng Zhu ,Mai Wang ,Charlotte R Pfeifer ,Yuntao Xia ,Steven Phan ,Jason C Andrechak ,Junhong Du ,Michael P Tobin ,Alisya Anlas ,Lawrence J Dooling ,Manasvita Vashisth ,Jerome Irianto ,Michael A Lampson ,Dennis E Discher

Physical Therapy for Gait, Balance, and Cognition in Individuals with Cognitive Impairment: A Retrospective Analysis

针对认知障碍患者的步态、平衡和认知功能的物理治疗:一项回顾性分析

Longhurst, Jason; Phan, Jason; Chen, Elbert; Jackson, Steven; Landers, Merrill R