日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Synthesis and Biological Evaluation of a Novel Dual-Targeting Small Molecule Drug Conjugate Modulating the Crosstalk between α5β1 Integrin and MDM2 in Glioblastoma

合成及生物学评价一种新型双靶点小分子药物偶联物，该偶联物可调节胶质母细胞瘤中α5β1整合素与MDM2之间的相互作用

期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00669
Arrigoni, Federico; Ferrari, Ana; Prpić, Helena; Markeviciute, Elena; Muzi, Alessia; Roscilli, Giuseppe; Gazzola, Silvia; Piarulli, Umberto
细胞生物学
MDM2
发表日期：2026
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Comparative Enzymatic and Stability Assays Reveal GPLG as an Effective Cathepsin B Cleavable Linker for Tumor-Targeting Drug Conjugates

酶学和稳定性比较分析表明，GPLG 是一种有效的组织蛋白酶 B 可裂解连接子，可用于肿瘤靶向药物偶联物。

期刊:ACS Omega
影响因子:4.3
doi:10.1021/acsomega.5c05758
Cazzaniga, Giulia; Zambra, Marco; Bongiolo, Samuele; Prpić, Helena; Fasola, Elettra; Arrigoni, Federico; Piarulli, Umberto; Gazzola, Silvia
肿瘤
肿瘤免疫
发表日期：2025
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Impairing protein-protein interactions in an essential tRNA modification complex: An innovative antimicrobial strategy against Pseudomonas aeruginosa

削弱必需的tRNA修饰复合物中的蛋白质-蛋白质相互作用：一种针对铜绿假单胞菌的创新抗菌策略

期刊:Journal of Peptide Science
影响因子:1.8
doi:10.1002/psc.3658
Bollati, Michela; Fasola, Elettra; Pieraccini, Stefano; Freddi, Francesca; Cocomazzi, Paolo; Oliva, Francesco; Klußmann, Merlin; Maspero, Angelo; Piarulli, Umberto; Ferrara, Silvia; Pellegrino, Sara; Bertoni, Giovanni; Gazzola, Silvia
发表日期：2025
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A combined fragment-based virtual screening and STD-NMR approach for the identification of E-cadherin ligands

一种结合基于片段的虚拟筛选和STD-NMR的E-钙黏蛋白配体鉴定方法

期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2022.946087
Vasile, Francesca; Lavore, Francesca; Gazzola, Silvia; Vettraino, Chiara; Parisini, Emilio; Piarulli, Umberto; Belvisi, Laura; Civera, Monica
发表日期：2022
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Conformational switch and multiple supramolecular structures of a newly identified self-assembling protein-mimetic peptide from Pseudomonas aeruginosa YeaZ protein

铜绿假单胞菌YeaZ蛋白中新发现的自组装蛋白模拟肽的构象转换和多种超分子结构

期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2022.1038796
Fasola, Elettra; Alboreggia, Giulia; Pieraccini, Stefano; Oliva, Francesco; Agharbaoui, Fatima Ezzahra; Bollati, Michela; Bertoni, Giovanni; Recchia, Sandro; Marelli, Marcello; Piarulli, Umberto; Pellegrino, Sara; Gazzola, Silvia
发表日期：2022
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Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

靶向血管内皮生长因子受体的抗血管生成螺旋寡肽的合理设计

期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2019.00170
Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano, Alvaro S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo
心血管
信号转导
血管生成
发表日期：2019
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Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α(V) β(3)

靶向整合素α(V)β(3)的RGD和isoDGR-单甲基奥瑞他汀缀合物的合成和生物学评价

期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.201900049
Raposo Moreira Dias, André; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkühler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto
发表日期：2019
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Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

隐藻素与RGD或isoDGR肽模拟物的偶联物用于靶向药物递送

期刊:ChemistryOpen
影响因子:3.1
doi:10.1002/open.201900110
Borbély, Adina; Figueras, Eduard; Martins, Ana; Bodero, Lizeth; Raposo Moreira Dias, André; López Rivas, Paula; Pina, Arianna; Arosio, Daniela; Gallinari, Paola; Frese, Marcel; Steinkühler, Christian; Gennari, Cesare; Piarulli, Umberto; Sewald, Norbert
发表日期：2019
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Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

RGD和isoDGR肽模拟物-α-鹅膏蕈碱缀合物的合成及生物学评价及其在肿瘤靶向治疗中的应用

期刊:Beilstein Journal of Organic Chemistry
影响因子:2.1
doi:10.3762/bjoc.14.29
Bodero, Lizeth; López Rivas, Paula; Korsak, Barbara; Hechler, Torsten; Pahl, Andreas; Müller, Christoph; Arosio, Daniela; Pignataro, Luca; Gennari, Cesare; Piarulli, Umberto
肿瘤免疫
肿瘤
发表日期：2018
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Insights into the Binding of Cyclic RGD Peptidomimetics to α(5)β(1) Integrin by using Live-Cell NMR And Computational Studies.

利用活细胞核磁共振和计算研究深入了解环状RGD肽模拟物与α(5)β(1)整合素的结合

期刊:ChemistryOpen
影响因子:3.1
doi:10.1002/open.201600112
Guzzetti Ileana, Civera Monica, Vasile Francesca, Arosio Daniela, Tringali Cristina, Piarulli Umberto, Gennari Cesare, Pignataro Luca, Belvisi Laura, Potenza Donatella
细胞生物学
发表日期：2017
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