日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Selective STING Activation in Intratumoral Myeloid Cells via CCR2-Directed Antibody-Drug Conjugate TAK-500

通过 CCR2 靶向抗体药物偶联物 TAK-500 选择性激活肿瘤内髓系细胞中的 STING

Vicky A Appleman ,Atsushi Matsuda ,Michelle L Ganno ,Dong Mei Zhang ,Emily Rosentrater ,Angel E Maldonado Lopez ,Angelo Porciuncula ,Tiquella Hatten ,Camilla L Christensen ,Samantha A Merrigan ,Hong Myung Lee ,Min Young Lee ,Charlotte I Wang ,Linlin Dong ,Jian Huang ,Natasha Iartchouk ,Jianing Wang ,He Xu ,Tomoki Yoneyama ,Konstantin I Piatkov ,Satyajeet Haridas ,Carole E Harbison ,Richard C Gregory ,Alexander Parent ,Neil Lineberry ,Chris Arendt ,Kurt A Schalper ,Adnan O Abu-Yousif

Identification of a Novel Linker Enabling the Bioconjugation of a Cyclic Dinucleotide for the STING Antibody-Drug Conjugate TAK-500

鉴定一种新型连接子,用于STING抗体-药物偶联物TAK-500的环状二核苷酸生物偶联

Lee, Hong Myung; Abdul-Hadi, Kojo; Appleman, Vicky A; Cardin, David; Dong, Linlin; England, Dylan; Ganno, Michelle L; Gershman, Rachel; Gigstad, Kenneth; Gulavita, Nanda; Hu, Zhigen; Huang, Jian; Huang, Shih-Chung; Lok, David; Ma, Liting; Malley, Jenna; Mizutani, Miho; Molchanova, Nina; Piatkov, Konstantin I; Rice, Elise; Shi, Zhan; Vyskocil, Stepan; Wang, Jianing; Xu, He; Xu, Tianlin; Zhang, Dong Mei; Zhang, Ji; Abu-Yousif, Adnan O

Quantifying LAGA mutated mouse IgG2a monoclonal antibody with a rapid pepsin digestion enabled immunoaffinity LC/MS/MS assay

使用快速胃蛋白酶消化免疫亲和 LC/MS/MS 分析法定量 LAGA 突变小鼠 IgG2a 单克隆抗体

Linlin Dong, Susan Chen, Konstantin Piatkov, Dong Wei, Mark G Qian

Leveraging a physiologically-based quantitative translational modeling platform for designing B cell maturation antigen-targeting bispecific T cell engagers for treatment of multiple myeloma

利用基于生理学的定量转化建模平台设计靶向B细胞成熟抗原的双特异性T细胞衔接器,用于治疗多发性骨髓瘤

Yoneyama, Tomoki; Kim, Mi-Sook; Piatkov, Konstantin; Wang, Haiqing; Zhu, Andy Z X

Downregulation of the Arg/N-degron Pathway Sensitizes Cancer Cells to Chemotherapy In Vivo

Arg/N-降解途径下调使癌细胞对体内化疗敏感

Dominique Leboeuf, Tatiana Abakumova, Tatiana Prikazchikova, Luke Rhym, Daniel G Anderson, Timofei S Zatsepin, Konstantin I Piatkov

The Arg/N-Degron Pathway-A Potential Running Back in Fine-Tuning the Inflammatory Response?

Arg/N-Degron 通路——微调炎症反应的潜在回跑者?

Dominique Leboeuf, Maxim Pyatkov, Timofei S Zatsepin, Konstantin Piatkov

Novel Apoptotic Mediators Identified by Conservation of Vertebrate Caspase Targets

通过脊椎动物半胱天冬酶靶点的保守性鉴定出新型凋亡介质

Gubina, Nina; Leboeuf, Dominique; Piatkov, Konstantin; Pyatkov, Maxim

Pharmacogenetics of anticancer monoclonal antibodies

抗癌单克隆抗体的药物遗传学

Shek, Dmitrii; Read, Scott A; Ahlenstiel, Golo; Piatkov, Irina

Beta-amyloid induces apoptosis of neuronal cells by inhibition of the Arg/N-end rule pathway proteolytic activity

β-淀粉样蛋白通过抑制Arg/N端规则通路蛋白水解活性诱导神经元细胞凋亡

Olga I Kechko, Irina Yu Petrushanko, Christopher S Brower, Alexei A Adzhubei, Alexey A Moskalev, Konstantin I Piatkov, Vladimir A Mitkevich, Alexander A Makarov

ABCB1 and ABCC1 single-nucleotide polymorphisms in patients treated with clozapine

接受氯氮平治疗的患者的 ABCB1 和 ABCC1 单核苷酸多态性

Irina Piatkov, Dorgival Caetano, Yolinda Assur, Sue Lynn Lau, Trudi Jones, Steven C Boyages, Mark McLean