日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of a Novel Linker Enabling the Bioconjugation of a Cyclic Dinucleotide for the STING Antibody-Drug Conjugate TAK-500

鉴定一种新型连接子,用于STING抗体-药物偶联物TAK-500的环状二核苷酸生物偶联

Lee, Hong Myung; Abdul-Hadi, Kojo; Appleman, Vicky A; Cardin, David; Dong, Linlin; England, Dylan; Ganno, Michelle L; Gershman, Rachel; Gigstad, Kenneth; Gulavita, Nanda; Hu, Zhigen; Huang, Jian; Huang, Shih-Chung; Lok, David; Ma, Liting; Malley, Jenna; Mizutani, Miho; Molchanova, Nina; Piatkov, Konstantin I; Rice, Elise; Shi, Zhan; Vyskocil, Stepan; Wang, Jianing; Xu, He; Xu, Tianlin; Zhang, Dong Mei; Zhang, Ji; Abu-Yousif, Adnan O

Leveraging a physiologically-based quantitative translational modeling platform for designing B cell maturation antigen-targeting bispecific T cell engagers for treatment of multiple myeloma

利用基于生理学的定量转化建模平台设计靶向B细胞成熟抗原的双特异性T细胞衔接器,用于治疗多发性骨髓瘤

Yoneyama, Tomoki; Kim, Mi-Sook; Piatkov, Konstantin; Wang, Haiqing; Zhu, Andy Z X

Novel Apoptotic Mediators Identified by Conservation of Vertebrate Caspase Targets

通过脊椎动物半胱天冬酶靶点的保守性鉴定出新型凋亡介质

Gubina, Nina; Leboeuf, Dominique; Piatkov, Konstantin; Pyatkov, Maxim

Analyzing N-terminal Arginylation through the Use of Peptide Arrays and Degradation Assays

利用肽阵列和降解分析法分析N端精氨酸化

Wadas, Brandon; Piatkov, Konstantin I; Brower, Christopher S; Varshavsky, Alexander

Formyl-methionine as a degradation signal at the N-termini of bacterial proteins.

甲酰甲硫氨酸作为细菌蛋白质 N 端的降解信号

Piatkov Konstantin I, Vu Tri T M, Hwang Cheol-Sang, Varshavsky Alexander

Calpain-generated natural protein fragments as short-lived substrates of the N-end rule pathway

钙蛋白酶生成的天然蛋白质片段作为N端规则途径的短寿命底物

Piatkov, Konstantin I; Oh, Jang-Hyun; Liu, Yuan; Varshavsky, Alexander

Ubiquitin reference technique and its use in ubiquitin-lacking prokaryotes.

泛素参考技术及其在缺乏泛素的原核生物中的应用

Piatkov Konstantin, Graciet Emmanuelle, Varshavsky Alexander

The N-end rule pathway counteracts cell death by destroying proapoptotic protein fragments

N端规则通路通过破坏促凋亡蛋白片段来对抗细胞死亡。

Piatkov, Konstantin I; Brower, Christopher S; Varshavsky, Alexander