日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nerandomilast as the first PDE4B-selective therapy in idiopathic pulmonary fibrosis

Nerandomilast 作为首个用于治疗特发性肺纤维化的 PDE4B 选择性疗法

Ibrahim, Md; Piazza, Gary A; Ahsan, Fakhrul

ADT-030, a novel PDE10 inhibitor, demonstrates potent antitumor activity in pancreatic ductal adenocarcinoma

ADT-030 是一种新型 PDE10 抑制剂,在胰腺导管腺癌中表现出强大的抗肿瘤活性。

Bandi, Dhana Sekhar Reddy; Nagaraju, Ganji Purnachandra; Sarvesh, Sujith; Foote, Jeremy B; Keeton, Adam B; Chen, Xi; Ramirez-Alcantara, Veronica; Holmes, Thomas; Akce, Mehmet; Singh, Anju; Powell, Craig M; Behera, Santosh; Azmi, Asfar S; Nurmemmedov, Elmar; Babic, Ivan; Gorman, Gregory S; Coward, Lori; Buchsbaum, Donald J; Maxuitenko, Yulia Y; Piazza, Gary A; El-Rayes, Bassel F

ADT-1004: a first-in-class, oral pan-RAS inhibitor with robust antitumor activity in preclinical models of pancreatic ductal adenocarcinoma

ADT-1004:一种首创的口服泛RAS抑制剂,在胰腺导管腺癌的临床前模型中具有强大的抗肿瘤活性

Bandi, Dhana Sekhar Reddy; Nagaraju, Ganji Purnachandra; Sarvesh, Sujith; Carstens, Julienne L; Foote, Jeremy B; Graff, Emily C; Fang, Yu-Hua D; Keeton, Adam B; Chen, Xi; Valiyaveettil, Jacob; Berry, Kristy L; Bae, Sejong; Akce, Mehmet; Gorman, Greg; Yoon, Karina J; Manne, Upender; Boyd, Michael R; Buchsbaum, Donald J; Azmi, Asfar S; Maxuitenko, Yulia Y; Piazza, Gary A; El-Rayes, Bassel F

Cyclic nucleotide phosphodiesterases as drug targets

环核苷酸磷酸二酯酶作为药物靶点

Kelly, Michy P; Nikolaev, Viacheslav O; Gobejishvili, Leila; Lugnier, Claire; Hesslinger, Christian; Nickolaus, Peter; Kass, David A; Pereira de Vasconcelos, Walma; Fischmeister, Rodolphe; Brocke, Stefan; Epstein, Paul M; Piazza, Gary A; Keeton, Adam B; Zhou, Gang; Abdel-Halim, Mohammad; Abadi, Ashraf H; Baillie, George S; Giembycz, Mark A; Bolger, Graeme; Snyder, Gretchen; Tasken, Kjetil; Saidu, Nathaniel E B; Schmidt, Martina; Zaccolo, Manuela; Schermuly, Ralph T; Ke, Hengming; Cote, Rick H; Mohammadi Jouabadi, Soroush; Roks, Anton J M

A Pan-RAS Inhibitor with a Unique Mechanism of Action Blocks Tumor Growth and Induces Antitumor Immunity in Gastrointestinal Cancer.

一种具有独特作用机制的泛 RAS 抑制剂可抑制肿瘤生长并诱导胃肠道癌症的抗肿瘤免疫

Foote Jeremy B, Mattox Tyler E, Keeton Adam B, Chen Xi, Smith Forrest T, Berry Kristy, Holmes Thomas W, Wang Junwei, Huang Chung-Hui, Ward Antonio, Mitra Amit K, Ramirez-Alcantara Veronica, Hardy Cherlene, Fleten Karianne G, Flatmark Kjersti, Yoon Karina J, Sarvesh Sujith, Nagaraju Ganji P, Bandi Dhana Sekhar Reddy, Maxuitenko Yulia Y, Valiyaveettil Jacob, Carstens Julienne L, Buchsbaum Donald J, Yang Jennifer, Zhou Gang, Nurmemmedov Elmar, Babic Ivan, Gaponeko Vadim, Abdelkarim Hazem, Boyd Michael R, Gorman Greg, Manne Upender, Bae Sejong, El-Rayes Bassel F, Piazza Gary A

Novel Disulfiram-Loaded Metal-Organic Nanoparticles Inhibit Tumor Growth and Induce Immunogenic Cell Death of Triple-Negative Breast Cancer Cells.

新型双硫仑负载金属有机纳米粒子抑制肿瘤生长并诱导三阴性乳腺癌细胞的免疫原性细胞死亡。

Huang Chung-Hui, Kang Xuejia, Zhou Lang, Wang Junwei, Wu Shuai, Sun Peizhen, Wang Qi, Keeton Adam B, Chen Pengyu, Piazza Gary A

Evaluation of a Novel Pan-RAS Inhibitor in 3D Bioprinted Tumor Models

在3D生物打印肿瘤模型中评估一种新型泛RAS抑制剂

De Nobrega, Daniela D; Eiler, Logan C; Ahirwar, Parmanand; Nallapu, Sonika; Rawal, Urvi P; Crawford, Chelsea L; Buchsbaum, Donald J; Keeton, Adam B; Maxuitenko, Yulia Y; Chen, Xi; Piazza, Gary A; Tsung, Allan; Budhwani, Karim I

Editorial: RAS inhibitor therapy of cancer

社论:RAS抑制剂治疗癌症

Buchsbaum, Donald J; Nassar, Nicolas N; Piazza, Gary A

Potency and selectivity of a novel pan-RAS inhibitor in 3D bioprinted organoid tumor models

新型泛RAS抑制剂在3D生物打印类器官肿瘤模型中的效力和选择性

De Nobrega, Daniela; Eiler, Logan C; Ahirwar, Parmanand; Rawal, Urvi P; Crawford, Chelsea L; Buchsbaum, Donald J; Keeton, Adam B; Maxuitenko, Yulia Y; Chen, Xi; Piazza, Gary A; Tsung, Allan; Budhwani, Karim I

Assessment of KRAS(G12C) inhibitors for colorectal cancer

评估KRAS(G12C)抑制剂在结直肠癌中的应用

Piazza, Gary A; Chandrasekaran, Preethi; Maxuitenko, Yulia Y; Budhwani, Karim I