日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Safety, Tolerability, Pharmacokinetics and Initial Pharmacodynamics of a Subcommissural Organ-Spondin-Derived Peptide: A Randomized, Placebo-Controlled, Double-Blind, Single Ascending Dose First-in-Human Study

下颌下器官-Spondin衍生肽的安全性、耐受性、药代动力学和初始药效学:一项随机、安慰剂对照、双盲、单次递增剂量首次人体研究

Bourdès, Valérie; Dogterom, Peter; Aleman, André; Parmantier, Pierre; Colas, Damien; Lemarchant, Sighild; Marie, Sébastien; Chou, Thomas; Abd-Elaziz, Khalid; Godfrin, Yann

Functional characterization of CDK10 and cyclin M truncated variants causing severe developmental disorders

导致严重发育障碍的 CDK10 和细胞周期蛋白 M 截短变体的功能表征

Thomas Robert, Anne-Catherine Dock-Bregeon, Pierre Colas

Kinase-Based Screening of Marine Natural Extracts Leads to the Identification of a Cytotoxic High Molecular Weight Metabolite from the Mediterranean Sponge Crambe tailliezi

基于激酶的海洋天然提取物筛选可鉴定出来自地中海海绵 Crambe tailliezi 的细胞毒性高分子量代谢物

Thi-Ngoc-Dung Nguyen, Omid Feizbakhsh, Estelle Sfecci, Blandine Baratte, Claire Delehouzé, Adrien Garcia, Corentin Moulin, Pierre Colas, Sandrine Ruchaud, Mohamed Mehiri, Stéphane Bach

A homozygous deleterious CDK10 mutation in a patient with agenesis of corpus callosum, retinopathy, and deafness

患有胼胝体发育不全、视网膜病变和耳聋的患者出现纯合有害 CDK10 突变

Vincent J Guen, Simon Edvardson, Nitay D Fraenkel, Aviva Fattal-Valevski, Chaim Jalas, Irene Anteby, Avraham Shaag, Talia Dor, David Gillis, Eitan Kerem, Jacqueline A Lees, Pierre Colas, Orly Elpeleg

STAR syndrome-associated CDK10/Cyclin M regulates actin network architecture and ciliogenesis

STAR 综合征相关 CDK10/Cyclin M 调节肌动蛋白网络结构和纤毛发生

Vincent J Guen, Carly Gamble, Dahlia E Perez, Sylvie Bourassa, Hildegard Zappel, Jutta Gärtner, Jacqueline A Lees, Pierre Colas

Spatially uniform enhancement of single quantum dot emission using plasmonic grating decoupler

利用等离子体光栅解耦器实现单个量子点发射的空间均匀增强

Kumar, Arunandan; Weeber, Jean-Claude; Bouhelier, Alexandre; Eloi, Fabien; Buil, Stéphanie; Quélin, Xavier; Nasilowski, Michel; Dubertret, Benoit; Hermier, Jean-Pierre; Colas des Francs, Gérard

Calcineurin A versus NS5A-TP2/HD domain containing 2: a case study of site-directed low-frequency random mutagenesis for dissecting target specificity of peptide aptamers

钙调神经磷酸酶 A 与 NS5A-TP2/HD 结构域 2:定点低频随机诱变案例研究,用于分析肽适体的靶向特异性

Silvia Dibenedetto, David Cluet, Pierre-Nicolas Stebe, Véronique Baumle, Jérémie Léault, Raphaël Terreux, Marc Bickle, Benoit D E Chassey, Ivan Mikaelian, Pierre Colas, Martin Spichty, Michele Zoli, Brian B Rudkin

CDK10/cyclin M is a protein kinase that controls ETS2 degradation and is deficient in STAR syndrome

CDK10/细胞周期蛋白 M 是一种控制 ETS2 降解的蛋白激酶,在 STAR 综合征中存在缺陷

Vincent J Guen, Carly Gamble, Marc Flajolet, Sheila Unger, Aurélie Thollet, Yoan Ferandin, Andrea Superti-Furga, Pascale A Cohen, Laurent Meijer, Pierre Colas

A RasGAP SH3 peptide aptamer inhibits RasGAP-Aurora interaction and induces caspase-independent tumor cell death

RasGAP SH3 肽适体抑制 RasGAP-Aurora 相互作用并诱导 caspase 非依赖性肿瘤细胞死亡

Perayot Pamonsinlapatham, Réda Hadj-Slimane, Françoise Raynaud, Marc Bickle, Claudine Corneloup, Audrey Barthelaix, Yves Lepelletier, Perrine Mercier, Matthieu Schapira, Jérôme Samson, Anne-Laure Mathieu, Nicolas Hugo, Olivier Moncorgé, Ivan Mikaelian, Sylvie Dufour, Christiane Garbay, Pierre Colas

Evidence for crucial electrostatic interactions between Bcl-2 homology domains BH3 and BH4 in the anti-apoptotic Nr-13 protein

抗凋亡 Nr-13 蛋白中 Bcl-2 同源域 BH3 和 BH4 之间存在关键静电相互作用的证据

Philippe Lalle, Abdel Aouacheria, Agnès Dumont-Miscopein, Martin Jambon, Séverine Venet, Hélène Bobichon, Pierre Colas, Gilbert Deléage, Christophe Geourjon, Germain Gillet