日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction

优化 Keap1-Nrf2 蛋白质-蛋白质相互作用的大环抑制剂时揭示结合位点水合和柔韧性的重要性

Fabio Begnini, Stefan Geschwindner, Patrik Johansson, Lisa Wissler, Richard J Lewis, Emma Danelius, Andreas Luttens, Pierre Matricon, Jens Carlsson, Stijn Lenders, Beate König, Anna Friedel, Peter Sjö, Stefan Schiesser, Jan Kihlberg

Agonist-induced dimer dissociation as a macromolecular step in G protein-coupled receptor signaling

激动剂诱导的二聚体解离是 G 蛋白偶联受体信号传导中的大分子步骤

Julian Petersen, Shane C Wright, David Rodríguez, Pierre Matricon, Noa Lahav, Aviv Vromen, Assaf Friedler, Johan Strömqvist, Stefan Wennmalm, Jens Carlsson, Gunnar Schulte

The tyrosine Y2502.39 in Frizzled 4 defines a conserved motif important for structural integrity of the receptor and recruitment of Disheveled

Frizzled 4 中的酪氨酸 Y2502.39 定义了一个保守基序,对于受体的结构完整性和 Disheveled 的募集非常重要

Katerina Strakova, Pierre Matricon, Chika Yokota, Elisa Arthofer, Ondrej Bernatik, David Rodriguez, Ernest Arenas, Jens Carlsson, Vitezslav Bryja, Gunnar Schulte