Structure-guided DOT1L probe optimization by label-free ligand displacement
通过无标记配体置换进行结构引导的 DOT1L 探针优化
期刊:ACS Chemical Biology
影响因子:3.5
doi:10.1021/cb500796d
Joanna S Yi, Alexander J Federation, Jun Qi, Sirano Dhe-Paganon, Michael Hadler, Xiang Xu, Roodolph St Pierre, Anthony C Varca, Lei Wu, Jason J Marineau, William B Smith, Amanda Souza, Emma J Chory, Scott A Armstrong, James E Bradner