日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Late-stage peptide modification with salicylaldehyde tag enhances affinity for nuclear factor-kappa B essential modulator

后期肽修饰用水杨醛标签增强了对核因子-κB必需调节剂的亲和力

Mason, Mattia; Peqini, Kaliroi; Uggeri, Federico; Rondelli, Diego; Sattin, Sara; Pignataro, Luca; Pellegrino, Sara; Belvisi, Laura; Scarpa, Edoardo; Bucci, Raffaella; Dal Corso, Alberto

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker

利用体外质谱法对带有蛋白酶可切割和酸不稳定连接子的抗体-瑞喹莫德偶联物进行生物分布分析

Bisbal Lopez, Lydia; Ravazza, Domenico; Bocci, Matilde; Zana, Aureliano; Principi, Lucrezia; Dakhel Plaza, Sheila; Galbiati, Andrea; Gilardoni, Ettore; Scheuermann, Jörg; Neri, Dario; Pignataro, Luca; Gennari, Cesare; Cazzamalli, Samuele; Dal Corso, Alberto

Visible Light-Promoted β-Functionalization of Carbonyl Compounds in the Presence of Organic Dyes

可见光促进有机染料存在下羰基化合物的β-官能化

Dolcini, Luigi; Gandini, Tommaso; Castiglioni, Riccardo; Bossi, Alberto; Penconi, Marta; Dal Corso, Alberto; Gennari, Cesare; Pignataro, Luca

Advanced Pyrrolidine-Carbamate Self-Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release

具有叔胺基团的先进吡咯烷-氨基甲酸酯自毁间隔基可诱导超快速循环药物释放

Dal Corso, Alberto; Frigoli, Margaux; Prevosti, Martina; Mason, Mattia; Bucci, Raffaella; Belvisi, Laura; Pignataro, Luca; Gennari, Cesare

Notch3 contributes to T-cell leukemia growth via regulation of the unfolded protein response

Notch3 通过调节未折叠蛋白反应促进 T 细胞白血病的生长

Maria Valeria Giuli, Giulia Diluvio, Eugenia Giuliani, Giulia Franciosa, Laura Di Magno, Maria Gemma Pignataro, Luca Tottone, Carmine Nicoletti, Zein Mersini Besharat, Giovanna Peruzzi, Maria Pelullo, Rocco Palermo, Gianluca Canettieri, Claudio Talora, Giulia d'Amati, Diana Bellavia, Isabella Screpa

Insight into GEBR-32a: Chiral Resolution, Absolute Configuration and Enantiopreference in PDE4D Inhibition

深入了解 GEBR-32a:PDE4D 抑制中的手性拆分、绝对构型和对映选择性

Cavalloro, Valeria; Russo, Katia; Vasile, Francesca; Pignataro, Luca; Torretta, Archimede; Donini, Stefano; Semrau, Marta S; Storici, Paola; Rossi, Daniela; Rapetti, Federica; Brullo, Chiara; Parisini, Emilio; Bruno, Olga; Collina, Simona

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

靶向血管内皮生长因子受体的抗血管生成螺旋寡肽的合理设计

Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano, Alvaro S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

中性粒细胞弹性蛋白酶促进连接子裂解和紫杉醇从整合素靶向缀合物中释放

Raposo Moreira Dias, André; Pina, Arianna; Dean, Amelia; Lerchen, Hans-Georg; Caruso, Michele; Gasparri, Fabio; Fraietta, Ivan; Troiani, Sonia; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α(V) β(3)

靶向整合素α(V)β(3)的RGD和isoDGR-单甲基奥瑞他汀缀合物的合成和生物学评价

Raposo Moreira Dias, André; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkühler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

RGD和isoDGR肽模拟物-α-鹅膏蕈碱缀合物的合成及生物学评价及其在肿瘤靶向治疗中的应用

Bodero, Lizeth; López Rivas, Paula; Korsak, Barbara; Hechler, Torsten; Pahl, Andreas; Müller, Christoph; Arosio, Daniela; Pignataro, Luca; Gennari, Cesare; Piarulli, Umberto