日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Allosteric activation of the glutamate receptor mGlu2 by the serotonin receptor 5-HT(2A)

血清素受体 5-HT(2A) 对谷氨酸受体 mGlu2 的变构激活

Gai, Siyu; Lin, Li; Meng, Jiyong; Wu, Yichen; Xue, Li; Xu, Chanjuan; Sun, Qian; Ricarte, Adrià; Dalton, James; Renault, Pedro; Giraldo, Jesús; Pin, Jean-Philippe; Rondard, Philippe; Liu, Jianfeng

Nanobody therapy rescues behavioural deficits of NMDA receptor hypofunction.

纳米抗体疗法可挽救 NMDA 受体功能低下引起的行为缺陷

Oosterlaken Mathieu, Rogliardo Angelina, Lipina Tatiana, Lafon Pierre-André, Tsitokana Mireille Elodie, Keck Mathilde, Cahuzac Héloïse, Prieu-Sérandon Pierre, Diem Séverine, Derieux Cécile, Camberlin Célia, Lafont Chrystel, Meyer Damien, Chames Patrick, Vandermoere Franck, Marin Philippe, Prézeau Laurent, Servent Denis, Salahpour Ali, Ramsey Amy J, Bécamel Carine, Pin Jean-Philippe, Kniazeff Julie, Rondard Philippe

Multi-faceted roles of β-arrestins in G protein-coupled receptor endocytosis

β-arrestin在G蛋白偶联受体内吞作用中的多重作用

Liu, Junke; Xue, Li; Ravier, Magalie A; Eshak, Floriane; Acher, Francine C; Goupil-Lamy, Anne; Cimadevila, Marta; Drube, Julia; Hoffmann, Carsten; Inoue, Asuka; Trinquet, Eric; Dupuis, Elodie; Prézeau, Laurent; Pin, Jean-Philippe; Rondard, Philippe

Triple Labeling Resolves a GPCR Intermediate State by Using Three-Color Single Molecule FRET

三重标记法利用三色单分子FRET解析GPCR中间态

Bonhomme, Léo; Bilgen, Ecenaz; Clerté, Caroline; Pin, Jean-Philippe; Rondard, Philippe; Margeat, Emmanuel; Lamb, Don C; Quast, Robert B

A modular click ligand-directed approach to label endogenous dopamine D(1) receptors in live cells.

一种模块化的点击配体导向方法,用于标记活细胞中的内源性多巴胺D(1)受体

Gómez-Santacana Xavier, Boutonnet Marin, Martínez-Juvés Carles, Cimadevila Marta, Catena Juanlo, Moutin Enora, Roux Thomas, Trinquet Eric, Lamarque Laurent, Perroy Julie, Prézeau Laurent, Zwier Jurriaan M, Pin Jean-Philippe, Llebaria Amadeu

Targeting the Brain with Single-Domain Antibodies: Greater Potential Than Stated So Far?

利用单域抗体靶向大脑:其潜力远超目前所言?

Tsitokana, Mireille Elodie; Lafon, Pierre-André; Prézeau, Laurent; Pin, Jean-Philippe; Rondard, Philippe

Structural basis of the activation of metabotropic glutamate receptor 3

代谢型谷氨酸受体3激活的结构基础

Fang, Wei; Yang, Fan; Xu, Chanjuan; Ling, Shenglong; Lin, Li; Zhou, Yingxin; Sun, Wenjing; Wang, Xiaomei; Liu, Peng; Rondard, Philippe; Shi, Pan; Pin, Jean-Philippe; Tian, Changlin; Liu, Jianfeng

Allosteric modulators enhance agonist efficacy by increasing the residence time of a GPCR in the active state

变构调节剂通过增加GPCR在活性状态下的停留时间来增强激动剂的效力。

Cao, Anne-Marinette; Quast, Robert B; Fatemi, Fataneh; Rondard, Philippe; Pin, Jean-Philippe; Margeat, Emmanuel

A nanobody activating metabotropic glutamate receptor 4 discriminates between homo- and heterodimers

激活代谢型谷氨酸受体4的纳米抗体能够区分同源二聚体和异源二聚体

Haubrich, Jordi; Font, Joan; Quast, Robert B; Goupil-Lamy, Anne; Scholler, Pauline; Nevoltris, Damien; Acher, Francine; Chames, Patrick; Rondard, Philippe; Prézeau, Laurent; Pin, Jean-Philippe

Allosteric ligands control the activation of a class C GPCR heterodimer by acting at the transmembrane interface.

变构配体通过作用于跨膜界面来控制 C 类 GPCR 异二聚体的激活

Liu Lei, Fan Zhiran, Rovira Xavier, Xue Li, Roux Salomé, Brabet Isabelle, Xin Mingxia, Pin Jean-Philippe, Rondard Philippe, Liu Jianfeng