Initial Pharmacological Characterization of a Major Hydroxy Metabolite of PF-5190457: Inverse Agonist Activity of PF-6870961 at the Ghrelin Receptor
PF-5190457 主要羟基代谢物的初步药理学表征:PF-6870961 对生长素释放肽受体的逆激动剂活性
期刊:Journal of Pharmacology and Experimental Therapeutics
影响因子:3.1
doi:10.1124/jpet.122.001393
Sara L Deschaine, Morten A Hedegaard, Claire L Pince, Mehdi Farokhnia, Jacob E Moose, Ingrid A Stock, Sravani Adusumalli, Fatemeh Akhlaghi, James L Hougland, Agnieszka Sulima, Kenner C Rice, George F Koob, Leandro F Vendruscolo, Birgitte Holst, Lorenzo Leggio