日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N-Branched Tricyclic Guanidines as Novel Melanocortin-3 Receptor Agonists and Melanocortin-4 Receptor Antagonists

N-支链三环胍类化合物作为新型黑皮质素-3受体激动剂和黑皮质素-4受体拮抗剂

Weirath, Nicholas A; Zajac, Jonathan W P; Donow, Haley M; Lavoi, Travis M; Pinilla, Clemencia; Santos, Radleigh G; Prajapati, Ritu; Speth, Robert; Ericson, Mark D; Sarupria, Sapna; Giulianotti, Marcello A; Haskell-Luevano, Carrie

Structure-activity relationship of pyrrolidine pentamine derivatives as inhibitors of the aminoglycoside 6'- N -acetyltransferase type Ib

吡咯烷五胺衍生物作为氨基糖苷6'-N-乙酰转移酶Ib型抑制剂的构效关系

Sklenicka, Jan; Tran, Tung; Ramirez, Maria S; Donow, Haley M; Magaña, Angel J; LaVoi, Travis; Mamun, Yasir; Chapagain, Prem; Santos, Radleigh; Pinilla, Clemencia; Giulianotti, Marc A; Tolmasky, Marcelo E

Antigen-driven CD8 (+) T cell clonal expansion is a prominent feature of MASH in humans and mice

抗原驱动的CD8(+)T细胞克隆扩增是人和小鼠MASH的一个显著特征。

Burtis, Abbigayl E C; DeNicola, Destiny M C; Ferguson, Megan E; Santos, Radleigh G; Pinilla, Clemencia; Kriss, Michael S; Orlicky, David J; Tamburini, Beth A Jirón; Gillen, Austin E; Burchill, Matthew A

Restoring susceptibility to aminoglycosides: identifying small molecule inhibitors of enzymatic inactivation

恢复对氨基糖苷类抗生素的敏感性:鉴定酶失活的小分子抑制剂

Magaña, Angel J; Sklenicka, Jan; Pinilla, Clemencia; Giulianotti, Marc; Chapagain, Prem; Santos, Radleigh; Ramirez, Maria Soledad; Tolmasky, Marcelo E

Beryllium-specific CD4+ T cells induced by chemokine neoantigens perpetuate inflammation

由趋化因子新抗原诱导的铍特异性CD4+ T细胞会加剧炎症反应。

Falta, Michael T; Crawford, Jeremy C; Tinega, Alex N; Landry, Laurie G; Crawford, Frances; Mack, Douglas G; Martin, Allison K; Atif, Shaikh M; Li, Li; Santos, Radleigh G; Nakayama, Maki; Kappler, John W; Maier, Lisa A; Thomas, Paul G; Pinilla, Clemencia; Fontenot, Andrew P

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign

通过高通量“无偏”筛选活动发现纳摩尔级黑素皮质素-3受体(MC3R)选择性小分子吡咯烷双环胍激动剂化合物

Doering, Skye R; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G; Lavoi, Travis M; Giulianotti, Marc A; Pinilla, Clemencia; Appel, Jon R; Houghten, Richard A; Ericson, Mark D; Haskell-Luevano, Carrie

A Randomized Double-Blind Placebo-Controlled Phase II Trial of Dendritic Cell Vaccine ICT-107 in Newly Diagnosed Patients with Glioblastoma

一项针对新诊断胶质母细胞瘤患者的树突状细胞疫苗 ICT-107 的随机、双盲、安慰剂对照 II 期试验

Wen, Patrick Y; Reardon, David A; Armstrong, Terri S; Phuphanich, Surasak; Aiken, Robert D; Landolfi, Joseph C; Curry, William T; Zhu, Jay-Jiguang; Glantz, Michael; Peereboom, David M; Markert, James M; LaRocca, Renato; O'Rourke, Donald M; Fink, Karen; Kim, Lyndon; Gruber, Michael; Lesser, Glenn J; Pan, Edward; Kesari, Santosh; Muzikansky, Alona; Pinilla, Clemencia; Santos, Radleigh G; Yu, John S

Correction: Methodological approach to the ex vivo expansion and detection of T. cruzi-specific T cells from chronic Chagas disease patients

更正:体外扩增和检测慢性恰加斯病患者体内克氏锥虫特异性T细胞的方法学方法

Acevedo, Gonzalo R; Longhi, Silvia A; Bunying, Alcinette; Sabri, Nazila; Atienza, Augusto; Zago, María P; Santos, Radleigh; Judkowski, Valeria A; Pinilla, Clemencia; Gómez, Karina A

Rapid scanning structure-activity relationships in combinatorial data sets: identification of activity switches

快速扫描组合数据集中的构效关系:活性开关的识别

Medina-Franco, José L; Edwards, Bruce S; Pinilla, Clemencia; Appel, Jon R; Giulianotti, Marc A; Santos, Radleigh G; Yongye, Austin B; Sklar, Larry A; Houghten, Richard A

Selective agonists and antagonists of formylpeptide receptors: duplex flow cytometry and mixture-based positional scanning libraries

甲酰肽受体的选择性激动剂和拮抗剂:双重流式细胞术和基于混合物的定位扫描库

Pinilla, Clemencia; Edwards, Bruce S; Appel, Jon R; Yates-Gibbins, Tina; Giulianotti, Marc A; Medina-Franco, Jose L; Young, Susan M; Santos, Radleigh G; Sklar, Larry A; Houghten, Richard A