日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Development of PROTACs Targeting the Moonlighting Enzyme Nicotinamide Phosphoribosyltransferase (NAMPT) for Breast Cancer Therapy

开发靶向多功能酶烟酰胺磷酸核糖转移酶 (NAMPT) 的 PROTAC 用于乳腺癌治疗

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01827
Galli, Ubaldina; Moro, Marianna; Balestrero, Federica Carolina; Colombo, Giorgia; Koten, Marco; Roncaglio, Benedetta; Genazzani, Armando A; Aprile, Silvio; Massarotti, Alberto; Orsomando, Giuseppe; Pirali, Tracey; Grolla, Ambra A
肿瘤
肿瘤免疫
乳腺癌
NAMPT
发表日期：2026
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Expanding the Scope of PROTACs: Opportunities and Challenges in Topical Delivery

拓展PROTAC的范围：专题递送的机遇与挑战

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01911
Gioiello, Laura; Di Martino, Rita Maria Concetta; Pirali, Tracey
发表日期：2025
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Versatile One-Pot Synthesis of Hydrophobic Tags by Multicomponent Reactions

利用多组分反应实现疏水标签的多功能一锅法合成

期刊:ACS Omega
影响因子:4.3
doi:10.1021/acsomega.4c09726
Balestrero, Federica Carolina; Gioiello, Laura; Goutsiou, Georgia; Sangaletti, Sabina; Di Martino, Rita Maria Concetta; Condorelli, Fabrizio; Grolla, Ambra A; Pirali, Tracey
发表日期：2025
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Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1.

鉴定一种抑制吲哚胺 2,3-双加氧酶 1 的酶促和非酶促功能的化合物

期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.4c00265
Panfili Eleonora, Rezzi Sarah Jane, Adamo Annalisa, Mazzoletti Daniele, Massarotti Alberto, Miggiano Riccardo, Fallarini Silvia, Ambrosino Sara, Coletti Alice, Molinaro Pasquale, Milella Michele, Paiella Salvatore, Macchiarulo Antonio, Ugel Stefano, Pirali Tracey, Pallotta Maria Teresa
信号转导
发表日期：2024
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Deuterium in drug discovery: progress, opportunities and challenges

药物研发中的氘：进展、机遇与挑战

期刊:Nature Reviews Drug Discovery
影响因子:101.8
doi:10.1038/s41573-023-00703-8
Di Martino, Rita Maria Concetta; Maxwell, Brad D; Pirali, Tracey
发表日期：2023
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An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline

多索茶碱中氘诱导的意外代谢转换

期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.2c00166
Aprile, Silvio; Colombo, Giorgia; Serafini, Marta; Di Paola, Rosanna; Pisati, Federica; Bhela, Irene Preet; Cuzzocrea, Salvatore; Grosa, Giorgio; Pirali, Tracey
代谢
发表日期：2022
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What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications

名称的意义何在？基于国际非专利名称（INN）出版物的药物命名和药物化学趋势

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c00181
Serafini, Marta; Cargnin, Sarah; Massarotti, Alberto; Tron, Gian Cesare; Pirali, Tracey; Genazzani, Armando A
发表日期：2021
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Tritylamine as an Ammonia Surrogate in the Ugi Reaction Provides Access to Unprecedented 5-Sulfamido Oxazoles Using Burgess-type Reagents

三苯甲基胺作为氨的替代物用于Ugi反应，利用Burgess型试剂可合成前所未有的5-磺酰胺基噁唑

期刊:Organic Letters
影响因子:5
doi:10.1021/acs.orglett.1c01002
Bhela, Irene Preet; Serafini, Marta; Del Grosso, Erika; Tron, Gian Cesare; Pirali, Tracey
发表日期：2021
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Essential Medicinal Chemistry of Essential Medicines

基本药物的基本药物化学

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.0c00415
Serafini, Marta; Cargnin, Sarah; Massarotti, Alberto; Pirali, Tracey; Genazzani, Armando A
发表日期：2020
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Moonlighting Proteins Are Important Players in Cancer Immunology

兼职蛋白在癌症免疫学中扮演重要角色

期刊:Frontiers in Immunology
影响因子:5.9
doi:10.3389/fimmu.2020.613069
Adamo, Annalisa; Frusteri, Cristina; Pallotta, Maria Teresa; Pirali, Tracey; Sartoris, Silvia; Ugel, Stefano
Immunology/Inflammation
肿瘤
肿瘤免疫
免疫/内分泌
发表日期：2020
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