日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Evaluation of Sodium Channel Blockers with Anti-invasive Activities in Medullary Thyroid Cancer

设计、合成和评价具有抗甲状腺髓样癌侵袭活性的钠通道阻滞剂

Pukkanasut, Piyasuda; Dutta, Shilpa; Whitt, Jason; Babu, Parvathy; Lopez-Charcas, Osbaldo; Anguheven-Ledezma, Tonantzin Guadalupe; Gomora, Juan Carlos; Jaskula-Sztul, Renata; Velu, Sadanandan E

Characterizing SSTR2 expression and modulation for targeted imaging and therapy in preclinical models of triple-negative breast cancer.

在三阴性乳腺癌的临床前模型中,对 SSTR2 表达和调控进行表征,以用于靶向成像和治疗

Lynch Shannon E, Crawford Corinne I, Houson Hailey A, Omweri James M, Pukkanasut Piyasuda, Gallegos Carlos A, Whitt Jason D, Jaskula-Sztul Renata, Lapi Suzanne E, Sorace Anna G

Polymer vesicles for the delivery of inhibitors of cariogenic biofilm

用于递送致龋生物膜抑制剂的聚合物囊泡

Ahirwar, Parmanand; Kozlovskaya, Veronika; Pukkanasut, Piyasuda; Nikishau, Pavel; Nealy, Sarah; Harber, Gregory; Michalek, Suzanne M; Antony, Linto; Wu, Hui; Kharlampieva, Eugenia; Velu, Sadanandan E

Therapeutic targeting of voltage-gated sodium channel Na(V)1.7 for cancer metastasis

以电压门控钠通道Na(V)1.7为靶点治疗癌症转移

Pukkanasut, Piyasuda; Jaskula-Sztul, Renata; Gomora, Juan Carlos; Velu, Sadanandan E

Hydrogel-Encapsulated Biofilm Inhibitors Abrogate the Cariogenic Activity of Streptococcus mutans

水凝胶包裹的生物膜抑制剂可消除变形链球菌的致龋活性

Ahirwar, Parmanand; Kozlovskaya, Veronika; Nijampatnam, Bhavitavya; Rojas, Edwin M; Pukkanasut, Piyasuda; Inman, Daniel; Dolmat, Maksim; Law, Anna C; Schormann, Norbert; Deivanayagam, Champion; Harber, Gregory J; Michalek, Suzanne M; Wu, Hui; Kharlampieva, Eugenia; Velu, Sadanandan E

Voltage-Gated Sodium Channel NaV1.7 Inhibitors with Potent Anticancer Activities in Medullary Thyroid Cancer Cells

电压门控钠通道 NaV1.7 抑制剂对髓样甲状腺癌细胞具有强效抗癌活性

Piyasuda Pukkanasut, Jason Whitt, Rachael Guenter, Shannon E Lynch, Carlos Gallegos, Margarita Jacaranda Rosendo-Pineda, Juan Carlos Gomora, Herbert Chen, Diana Lin, Anna Sorace, Renata Jaskula-Sztul, Sadanandan E Velu

Voltage-Gated Sodium Channel NaV1.5 Controls NHE-1-Dependent Invasive Properties in Colon Cancer Cells

电压门控钠通道 NaV1.5 控制结肠癌细胞中的 NHE-1 依赖性侵袭特性

Osbaldo Lopez-Charcas, Lucile Poisson, Oumnia Benouna, Roxane Lemoine, Stéphanie Chadet, Adrien Pétereau, Widad Lahlou, Serge Guyétant, Mehdi Ouaissi, Piyasuda Pukkanasut, Shilpa Dutta, Sadanandan E Velu, Pierre Besson, Driffa Moussata, Sébastien Roger

Pharmacological and nutritional targeting of voltage-gated sodium channels in the treatment of cancers

癌症治疗中电压门控钠通道的药理学和营养学靶向治疗

Lopez-Charcas, Osbaldo; Pukkanasut, Piyasuda; Velu, Sadanandan E; Brackenbury, William J; Hales, Tim G; Besson, Pierre; Gomora, Juan Carlos; Roger, Sébastien

Discovery of Potent Inhibitors of Streptococcus mutans Biofilm with Antivirulence Activity

发现具有抗毒力活性的强效变形链球菌生物膜抑制剂

Nijampatnam, Bhavitavya; Ahirwar, Parmanand; Pukkanasut, Piyasuda; Womack, Holly; Casals, Luke; Zhang, Hua; Cai, Xia; Michalek, Suzanne M; Wu, Hui; Velu, Sadanandan E