Palazestrant, a novel oral Complete Estrogen Receptor Antagonist (CERAN) and Selective Estrogen Receptor Degrader (SERD), in patients with ER+/HER2- advanced or metastatic breast cancer: phase 1/2 study results
帕拉塞群(Palazestrant)是一种新型口服完全雌激素受体拮抗剂(CERAN)和选择性雌激素受体降解剂(SERD),用于治疗ER+/HER2-晚期或转移性乳腺癌患者:1/2期研究结果
期刊:Breast Cancer Research
影响因子:5.6
doi:10.1186/s13058-025-02049-y
Hamilton, Erika P; Patel, Manish R; Borges, Virginia F; Meisel, Jane L; Okera, Meena; Alemany, Carlos A; Pluard, Timothy J; Wesolowski, Robert; Sabanathan, Dhanusha; Miller, Kathy D; Conlin, Alison K; McCarthy, Nicole; Shaw, Morena; Tonda, Margaret; Shilkrut, Mark; Lin, Nancy U
肿瘤
HER2
肿瘤免疫
RAN
信号转导
乳腺癌
免疫/内分泌