日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Author Correction: Regulation of nucleotide metabolism by mutant p53 contributes to its gain-of-function activities

作者更正:突变型p53对核苷酸代谢的调控有助于其获得功能活性。

Kollareddy, Madhusudhan; Dimitrova, Elizabeth; Vallabhaneni, Krishna C; Chan, Adriano; Le, Thuc; Chauhan, Krishna M; Carrero, Zunamys I; Ramakrishnan, Gopalakrishnan; Watabe, Kounosuke; Haupt, Ygal; Haupt, Sue; Pochampally, Radhika; Boss, Gerard R; Romero, Damian G; Radu, Caius G; Martinez, Luis A

Discovery of potent and brain-penetrable tubulin inhibitors that effectively suppress breast cancer brain metastasis.

发现强效且能穿透血脑屏障的微管蛋白抑制剂,可有效抑制乳腺癌脑转移。

Krutilina Raisa I, Adeleye Kelli L, Playa Hilaire C, Pochampally Satyanarayana, Banjeree Souvik, Oluwalana Damilola, Kamal Mir Shahriar, Tian Di, Miller Duane D, Li Wei, Seagroves Tiffany N

Structural Activity Relationship Analysis of New Diphenyl PFI-3 Analogues Targeting for the Treatment of Glioblastoma

针对胶质母细胞瘤治疗的新型二苯基PFI-3类似物的结构活性关系分析

Hwang, Dong-Jin; Yang, Chuanhe; Wang, Yinan; Kelso, Hannah; Pochampally, Satyanarayana; Pfeffer, Lawrence M; Miller, Duane D

A Pyrimidine-Based Tubulin Inhibitor Shows Potent Anti-Glioblastoma Activity In Vitro and In Vivo

一种基于嘧啶的微管蛋白抑制剂在体外和体内均显示出强大的抗胶质母细胞瘤活性

Pochampally, Satyanarayana; Pfeffer, Lawrence M; Miranda-Carboni, Gustavo A; Daniel, Macey; James, Jazz I; Smith, Allana; Yang, Chuan He; Kelso, Hannah R; Parke, Deanna N; Hwang, Dong-Jin; Li, Wei; Miller, Duane D

Novel Antimitotic Agent SP-1-39 Inhibits Head and Neck Squamous Cell Carcinoma.

新型抗有丝分裂剂 SP-1-39 可抑制头颈部鳞状细胞癌

Adeleye K L, Li A R, Xie Y, Pochampally S, Hamilton D, Garcia-Godoy F, Miller D D, Li W

SB226, an inhibitor of tubulin polymerization, inhibits paclitaxel-resistant melanoma growth and spontaneous metastasis

SB226 是一种微管蛋白聚合抑制剂,可抑制紫杉醇耐药性黑色素瘤的生长和自发转移

Shanshan Deng, Souvik Banerjee, Hao Chen, Satyanarayana Pochampally, Yuxi Wang, Mi-Kyung Yun, Stephen W White, Keyur Parmar, Bernd Meibohm, Kelli L Hartman, Zhongzhi Wu, Duane D Miller, Wei Li

Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo

嘧啶二氢喹喔啉酮衍生物的设计、合成和生物学评价作为微管蛋白秋水仙碱位点结合剂,在体外和体内均表现出有效的抗癌活性

Satyanarayana Pochampally, Kelli L Hartman, Rui Wang, Jiaxing Wang, Mi-Kyung Yun, Keyur Parmar, Hyunseo Park, Bernd Meibohm, Stephen W White, Wei Li, Duane D Miller

Synthesis, antimicrobial and antioxidant activity of triazole, pyrazole containing thiazole derivatives and molecular docking studies on COVID-19

三唑、吡唑类噻唑衍生物的合成、抗菌和抗氧化活性研究及其对新冠病毒的分子对接研究

Matta, Raghavender; Pochampally, Jalapathi; Dhoddi, Bala Narsimha; Bhookya, Shankar; Bitla, Sampath; Akkiraju, Anjini Gayatri

Polycomb group protein Suz12 is regulated by a novel miRNA-like small RNA

Polycomb 组蛋白 Suz12 受新型 miRNA 样小 RNA 调控

Patrice Penfornis, Joseph D Fernandes, Radhika R Pochampally

Synthesis, anti-microbial activity, cytotoxicity of some novel substituted (5-(3-(1H-benzo[d]imidazol-2-yl)-4-hydroxybenzyl)benzofuran-2-yl)(phenyl)methanone analogs

一些新型取代的(5-(3-(1H-苯并[d]咪唑-2-基)-4-羟基苄基)苯并呋喃-2-基)(苯基)甲酮类似物的合成、抗菌活性和细胞毒性

Bhookya Shankar, Pochampally Jalapathi, Balabadra Saikrishna, Shaym Perugu, Vijjulatha Manga