日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulphostin-inspired N-phosphonopiperidones as selective covalent DPP8 and DPP9 inhibitors.

受磺基膦酸酯启发而合成的 N-膦酸哌啶酮类化合物作为选择性共价 DPP8 和 DPP9 抑制剂

Sewald Leonard, Tabak Werner W A, Fehr Lorenz, Zolg Samuel, Najdzion Maja, Verhoef Carlo J A, Podlesainski David, Geiss-Friedlander Ruth, Lammens Alfred, Kaschani Farnusch, Hellerschmied Doris, Huber Robert, Kaiser Markus

Structure function analysis of ADP-dependent cyanobacterial phosphofructokinase reveals new phylogenetic grouping in the PFK-A family.

对 ADP 依赖性蓝细菌磷酸果糖激酶的结构功能分析揭示了 PFK-A 家族中新的系统发育分组

Shen Lu, Peraglie Carmen, Podlesainski David, Stracke Christina, Ojha Ravi Shankar, Caliebe Frauke, Kaiser Markus, Forchhammer Karl, Hagemann Martin, Gutekunst Kirstin, Snoep Jacky L, Bräsen Christopher, Siebers Bettina

Chemoproteomics-Enabled Identification of 4-Oxo-β-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9

化学蛋白质组学鉴定4-氧代-β-内酰胺类化合物作为二肽基肽酶8和9的抑制剂

Carvalho, Luís A R; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Wöhrle, Svenja; Lum, Kenneth M; Podlesainski, David; Vieira, Andreia C; Kiefersauer, Reiner; Félix, Rita; Rodrigues, Tiago; Lucas, Susana D; Groß, Olaf; Geiss-Friedlander, Ruth; Cravatt, Benjamin F; Huber, Robert; Kaiser, Markus; Moreira, Rui