日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nitroreductase-triggered indazole formation

硝基还原酶触发的吲唑形成

Terholsen, Henrik; Medema, Lisa; Chernyshova, Elizaveta; Prats Luján, Alejandro; Poelarends, Gerrit J; Schmidt, Sandy

Asymmetric Conjugate Hydrocyanation of α,β-Unsaturated Aldehydes Catalyzed by Engineered 2-Deoxy-D-ribose-5-phosphate Aldolase

工程改造的2-脱氧-D-核糖-5-磷酸醛缩酶催化α,β-不饱和醛的不对称共轭氢氰化反应

Zhou, Hangyu; Fodran, Peter; Fu, Haigen; Poelarends, Gerrit J

Engineered C-N Lyases for Stereoselective Synthesis of Tertiary Amines

工程化CN裂解酶用于立体选择性合成叔胺

Bothof, Laura; Gong, Xiaofang; Onclin, Marrit E; Fodran, Peter; Poelarends, Gerrit J

Engineering 2-Deoxy-D-ribose-5-phosphate Aldolase for anti- and syn-Selective Epoxidations of α,β-Unsaturated Aldehydes

工程改造 2-脱氧-D-核糖-5-磷酸醛缩酶用于 α,β-不饱和醛的反式和顺式选择性环氧化反应

Zhou, Hangyu; Kunzendorf, Andreas; Xu, Guangcai; Frietema, Hylke O T; Thunnissen, Andy-Mark W H; Poelarends, Gerrit J

Correction to "Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione Derivative Inhibits d-Dopachrome Tautomerase Activity and Suppresses the Proliferation of Non-Small Cell Lung Cancer Cells"

更正“噻吩并[2,3-d]嘧啶-2,4(1H,3H)-二酮衍生物抑制d-多巴色素互变酶活性并抑制非小细胞肺癌细胞增殖”

Xiao, Zhangping; Osipyan, Angelina; Song, Shanshan; Chen, Deng; Schut, Reinder A; van Merkerk, Ronald; van der Wouden, Petra E; Cool, Robbert H; Quax, Wim J; Melgert, Barbro N; Poelarends, Gerrit J; Dekker, Frank J

Multigram-scale chemoenzymatic synthesis of diverse aminopolycarboxylic acids as potential metallo-β-lactamase inhibitors

多克级化学酶法合成多种氨基多羧酸作为潜在的金属β-内酰胺酶抑制剂

Bhat, Mohammad Faizan; Prats Luján, Alejandro; Saifuddin, Mohammad; Fodran, Peter; Poelarends, Gerrit J

Allosteric Inhibitors of Macrophage Migration Inhibitory Factor (MIF) Interfere with Apoptosis-Inducing Factor (AIF) Co-Localization to Prevent Parthanatos.

巨噬细胞迁移抑制因子 (MIF) 的变构抑制剂干扰凋亡诱导因子 (AIF) 的共定位,从而阻止细胞凋亡

Chen Deng, Osipyan Angelina, Adriana Jeaunice, Kader Mohammed, Gureev Maxim, Knol Catharina W J, Sigmund Marie-Cathérine, Xiao Zhangping, van der Wouden Petra E, Cool Robbert H, Poelarends Gerrit J, Dekker Frank J

Gene Fusion and Directed Evolution to Break Structural Symmetry and Boost Catalysis by an Oligomeric C-C Bond-Forming Enzyme

基因融合和定向进化打破结构对称性并增强寡聚C-C键形成酶的催化活性

Xu, Guangcai; Kunzendorf, Andreas; Crotti, Michele; Rozeboom, Henriëtte J; Thunnissen, Andy-Mark W H; Poelarends, Gerrit J

Unlocking New Reactivities in Enzymes by Iminium Catalysis

利用亚胺催化释放酶的新反应活性

Xu, Guangcai; Poelarends, Gerrit J

Chemoenzymatic Asymmetric Synthesis of Complex Heterocycles: Dihydrobenzoxazinones and Dihydroquinoxalinones

复杂杂环化合物的化学酶法不对称合成:二氢苯并噁嗪酮和二氢喹喔啉酮

Bhat, Mohammad Faizan; Luján, Alejandro Prats; Saifuddin, Mohammad; Poelarends, Gerrit J