日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CU Cilia - an application for image analysis by machine learning - reveals significance of cysteine cathepsin K activity for primary cilia of human thyroid epithelial cells

CU Cilia——一款基于机器学习的图像分析应用程序——揭示了半胱氨酸蛋白酶K活性对人甲状腺上皮细胞原纤毛的重要性

Rehders, Maren; Alekseitseva, Kseniia; Gissoni, João; Doğru, Alara G; Popov, Petr; Boiarov, Andrei; Brix, Klaudia

OrgNet: orientation-gnostic protein stability assessment using convolutional neural networks

OrgNet:基于卷积神经网络的与方向无关的蛋白质稳定性评估

Buyanov, Ilya; Sarycheva, Anastasia; Popov, Petr

Structural insights into the high basal activity and inverse agonism of the orphan receptor GPR6 implicated in Parkinson's disease.

帕金森病中孤儿受体 GPR6 的高基础活性和反向激动作用的结构见解

Barekatain Mahta, Johansson Linda C, Lam Jordy H, Chang Hao, Sadybekov Anastasiia V, Han Gye Won, Russo Joseph, Bliesath Joshua, Brice Nicola L, Carlton Mark B L, Saikatendu Kumar S, Sun Hukai, Murphy Sean T, Monenschein Holger, Schiffer Hans H, Popov Petr, Lutomski Corinne A, Robinson Carol V, Liu Zhi-Jie, Hua Tian, Katritch Vsevolod, Cherezov Vadim

Approaching Optimal pH Enzyme Prediction with Large Language Models

利用大型语言模型预测最佳pH酶活性

Zaretckii, Mark; Buslaev, Pavel; Kozlovskii, Igor; Morozov, Alexander; Popov, Petr

A community effort in SARS-CoV-2 drug discovery

社区在SARS-CoV-2药物研发方面的努力

Schimunek, Johannes; Seidl, Philipp; Elez, Katarina; Hempel, Tim; Le, Tuan; Noé, Frank; Olsson, Simon; Raich, Lluís; Winter, Robin; Gokcan, Hatice; Gusev, Filipp; Gutkin, Evgeny M; Isayev, Olexandr; Kurnikova, Maria G; Narangoda, Chamali H; Zubatyuk, Roman; Bosko, Ivan P; Furs, Konstantin V; Karpenko, Anna D; Kornoushenko, Yury V; Shuldau, Mikita; Yushkevich, Artsemi; Benabderrahmane, Mohammed B; Bousquet-Melou, Patrick; Bureau, Ronan; Charton, Beatrice; Cirou, Bertrand C; Gil, Gérard; Allen, William J; Sirimulla, Suman; Watowich, Stanley; Antonopoulos, Nick; Epitropakis, Nikolaos; Krasoulis, Agamemnon; Itsikalis, Vassilis; Theodorakis, Stavros; Kozlovskii, Igor; Maliutin, Anton; Medvedev, Alexander; Popov, Petr; Zaretckii, Mark; Eghbal-Zadeh, Hamid; Halmich, Christina; Hochreiter, Sepp; Mayr, Andreas; Ruch, Peter; Widrich, Michael; Berenger, Francois; Kumar, Ashutosh; Yamanishi, Yoshihiro; Zhang, Kam Y J; Bengio, Emmanuel; Bengio, Yoshua; Jain, Moksh J; Korablyov, Maksym; Liu, Cheng-Hao; Marcou, Gilles; Glaab, Enrico; Barnsley, Kelly; Iyengar, Suhasini M; Ondrechen, Mary Jo; Haupt, V Joachim; Kaiser, Florian; Schroeder, Michael; Pugliese, Luisa; Albani, Simone; Athanasiou, Christina; Beccari, Andrea; Carloni, Paolo; D'Arrigo, Giulia; Gianquinto, Eleonora; Goßen, Jonas; Hanke, Anton; Joseph, Benjamin P; Kokh, Daria B; Kovachka, Sandra; Manelfi, Candida; Mukherjee, Goutam; Muñiz-Chicharro, Abraham; Musiani, Francesco; Nunes-Alves, Ariane; Paiardi, Giulia; Rossetti, Giulia; Sadiq, S Kashif; Spyrakis, Francesca; Talarico, Carmine; Tsengenes, Alexandros; Wade, Rebecca C; Copeland, Conner; Gaiser, Jeremiah; Olson, Daniel R; Roy, Amitava; Venkatraman, Vishwesh; Wheeler, Travis J; Arthanari, Haribabu; Blaschitz, Klara; Cespugli, Marco; Durmaz, Vedat; Fackeldey, Konstantin; Fischer, Patrick D; Gorgulla, Christoph; Gruber, Christian; Gruber, Karl; Hetmann, Michael; Kinney, Jamie E; Padmanabha Das, Krishna M; Pandita, Shreya; Singh, Amit; Steinkellner, Georg; Tesseyre, Guilhem; Wagner, Gerhard; Wang, Zi-Fu; Yust, Ryan J; Druzhilovskiy, Dmitry S; Filimonov, Dmitry A; Pogodin, Pavel V; Poroikov, Vladimir; Rudik, Anastassia V; Stolbov, Leonid A; Veselovsky, Alexander V; De Rosa, Maria; De Simone, Giada; Gulotta, Maria R; Lombino, Jessica; Mekni, Nedra; Perricone, Ugo; Casini, Arturo; Embree, Amanda; Gordon, D Benjamin; Lei, David; Pratt, Katelin; Voigt, Christopher A; Chen, Kuang-Yu; Jacob, Yves; Krischuns, Tim; Lafaye, Pierre; Zettor, Agnès; Rodríguez, M Luis; White, Kris M; Fearon, Daren; Von Delft, Frank; Walsh, Martin A; Horvath, Dragos; Brooks, Charles L 3rd; Falsafi, Babak; Ford, Bryan; García-Sastre, Adolfo; Yup Lee, Sang; Naffakh, Nadia; Varnek, Alexandre; Klambauer, Günter; Hermans, Thomas M

Molecular mechanism of biased signaling at the kappa opioid receptor.

kappa阿片受体偏向性信号传导的分子机制

El Daibani Amal, Paggi Joseph M, Kim Kuglae, Laloudakis Yianni D, Popov Petr, Bernhard Sarah M, Krumm Brian E, Olsen Reid H J, Diberto Jeffrey, Carroll F Ivy, Katritch Vsevolod, Wünsch Bernhard, Dror Ron O, Che Tao

Biphenyl scaffold for the design of NMDA-receptor negative modulators: molecular modeling, synthesis, and biological activity

联苯骨架用于设计NMDA受体负调控剂:分子建模、合成和生物活性

Karlov, Dmitry S; Temnyakova, Nadezhda S; Vasilenko, Dmitry A; Barygin, Oleg I; Dron, Mikhail Y; Zhigulin, Arseniy S; Averina, Elena B; Grishin, Yuri K; Grigoriev, Vladimir V; Gabrel'yan, Alexey V; Aniol, Viktor A; Gulyaeva, Natalia V; Osipenko, Sergey V; Kostyukevich, Yury I; Palyulin, Vladimir A; Popov, Petr A; Fedorov, Maxim V

Structure-based deep learning for binding site detection in nucleic acid macromolecules

基于结构的深度学习在核酸大分子结合位点检测中的应用

Kozlovskii, Igor; Popov, Petr

Spatiotemporal identification of druggable binding sites using deep learning

利用深度学习进行药物结合位点的时空识别

Kozlovskii, Igor; Popov, Petr

The structural study of mutation-induced inactivation of human muscarinic receptor M4

人类毒蕈碱受体M4突变诱导失活的结构研究

Wang, Jingjing; Wu, Meng; Wu, Lijie; Xu, Yueming; Li, Fei; Wu, Yiran; Popov, Petr; Wang, Lin; Bai, Fang; Zhao, Suwen; Liu, Zhi-Jie; Hua, Tian