日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ammonia Suppresses the Antitumor Activity of Natural Killer Cells and T Cells by Decreasing Mature Perforin.

氨通过减少成熟穿孔素来抑制自然杀伤细胞和T细胞的抗肿瘤活性

Domagala Joanna, Grzywa Tomasz M, Baranowska Iwona, Justyniarska Magdalena, Tannir Ryan, Graczyk-Jarzynka Agnieszka, Kusowska Aleksandra, Lecka Maria, Poreba Marcin, Fidyt Klaudyna, Marhelava Katsiaryna, Pilch Zofia, Picard Lea K, Wegierski Tomasz, Jastrzebski Kamil, Krawczyk Marta, Klopotowska Marta, Granica Monika, Urlaub Doris, Hajduk Szymon, Neeser Alexandra, Moros Spencer, Kozlowski Pawel, Bobrowicz Malgorzata, Miaczynska Marta, Ma Leyuan, Watzl Carsten, Winiarska Magdalena

Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin.

利用蛋白酶底物特异性筛选合理设计含非天然氨基酸的选择性蛋白酶抑制剂:应用于 HGFA、matriptase 和 hepsin

Mahoney Matthew W, Helander Jonathan, Kooner Anoopjit S, Norman Mariah, Damalanka Vishnu C, De Bona Paolo, Kasperkiewicz Paulina, Rut Wioletta, Poreba Marcin, Kashipathy Maithri M, Battaile Kevin P, Lovell Scott, O'Donoghue Anthony J, Craik Charles S, Drag Marcin, Janetka James W

Engineering caspase 7 as an affinity reagent to capture proteolytic products

将 caspase 7 改造为亲和试剂以捕获蛋白水解产物

Razai, Amir S; Snipas, Scott J; Poreba, Marcin; Fasci, Domenico; Salvesen, Guy S

Insights into ClpXP proteolysis: heterooligomerization and partial deactivation enhance chaperone affinity and substrate turnover in Listeria monocytogenes

对ClpXP蛋白水解的深入研究:异源寡聚化和部分失活增强单核细胞增生李斯特菌中分子伴侣的亲和力和底物周转率

Balogh, Dóra; Dahmen, Maria; Stahl, Matthias; Poreba, Marcin; Gersch, Malte; Drag, Marcin; Sieber, Stephan A

Emerging challenges in the design of selective substrates, inhibitors and activity-based probes for indistinguishable proteases

针对难以区分的蛋白酶,设计选择性底物、抑制剂和活性探针面临着新的挑战

Kasperkiewicz, Paulina; Poreba, Marcin; Groborz, Katarzyna; Drag, Marcin

Counter Selection Substrate Library Strategy for Developing Specific Protease Substrates and Probes.

反向选择底物库策略用于开发特异性蛋白酶底物和探针

Poreba Marcin, Solberg Rigmor, Rut Wioletta, Lunde Ngoc Nguyen, Kasperkiewicz Paulina, Snipas Scott J, Mihelic Marko, Turk Dusan, Turk Boris, Salvesen Guy S, Drag Marcin

Small Molecule Active Site Directed Tools for Studying Human Caspases

用于研究人类半胱天冬酶的小分子活性位点靶向工具

Poreba, Marcin; Szalek, Aleksandra; Kasperkiewicz, Paulina; Rut, Wioletta; Salvesen, Guy S; Drag, Marcin

Substrate Specificity and Possible Heterologous Targets of Phytaspase, a Plant Cell Death Protease

植物细胞死亡蛋白酶 Phytaspase 的底物特异性和可能的异源靶标

Raisa A Galiullina, Paulina Kasperkiewicz, Nina V Chichkova, Aleksandra Szalek, Marina V Serebryakova, Marcin Poreba, Marcin Drag, Andrey B Vartapetian

Caspase substrates and inhibitors

半胱天冬酶底物和抑制剂

Poreba, Marcin; Strózyk, Aleksandra; Salvesen, Guy S; Drag, Marcin

Probing the S1 specificity pocket of the aminopeptidases that generate antigenic peptides

探测产生抗原肽的氨肽酶的S1特异性口袋

Zervoudi, Efthalia; Papakyriakou, Athanasios; Georgiadou, Dimitra; Evnouchidou, Irini; Gajda, Anna; Poreba, Marcin; Salvesen, Guy S; Drag, Marcin; Hattori, Akira; Swevers, Luc; Vourloumis, Dionisios; Stratikos, Efstratios