日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological restoration of GTP hydrolysis by mutant RAS

突变RAS对GTP水解的药理恢复

Antonio Cuevas-Navarro #, Yasin Pourfarjam #, Feng Hu, Diego J Rodriguez, Alberto Vides, Ben Sang, Shijie Fan, Yehuda Goldgur, Elisa de Stanchina, Piro Lito

Pan-KRAS inhibitor disables oncogenic signalling and tumour growth

泛 KRAS 抑制剂可抑制致癌信号传导和肿瘤生长

Dongsung Kim #, Lorenz Herdeis #, Dorothea Rudolph #, Yulei Zhao, Jark Böttcher, Alberto Vides, Carlos I Ayala-Santos, Yasin Pourfarjam, Antonio Cuevas-Navarro, Jenny Y Xue, Andreas Mantoulidis, Joachim Bröker, Tobias Wunberg, Otmar Schaaf, Johannes Popow, Bernhard Wolkerstorfer, Katrin Gabriele Kro

Chemical remodeling of a cellular chaperone to target the active state of mutant KRAS

通过化学方法改造细胞伴侣蛋白,使其靶向突变型KRAS的活性状态

Schulze, Christopher J; Seamon, Kyle J; Zhao, Yulei; Yang, Yu C; Cregg, Jim; Kim, Dongsung; Tomlinson, Aidan; Choy, Tiffany J; Wang, Zhican; Sang, Ben; Pourfarjam, Yasin; Lucas, Jessica; Cuevas-Navarro, Antonio; Ayala-Santos, Carlos; Vides, Alberto; Li, Chuanchuan; Marquez, Abby; Zhong, Mengqi; Vemulapalli, Vidyasiri; Weller, Caroline; Gould, Andrea; Whalen, Daniel M; Salvador, Anthony; Milin, Anthony; Saldajeno-Concar, Mae; Dinglasan, Nuntana; Chen, Anqi; Evans, Jim; Knox, John E; Koltun, Elena S; Singh, Mallika; Nichols, Robert; Wildes, David; Gill, Adrian L; Smith, Jacqueline A M; Lito, Piro

ATP enhances the error-prone ribonucleotide incorporation by the SARS-CoV-2 RNA polymerase

ATP 会增强 SARS-CoV-2 RNA 聚合酶对核糖核苷酸的易错掺入。

Pourfarjam, Yasin; Ma, Zhijun; Kim, In-Kwon

An atypical BRCT-BRCT interaction with the XRCC1 scaffold protein compacts human DNA Ligase IIIα within a flexible DNA repair complex

BRCT-BRCT 与 XRCC1 支架蛋白的非典型相互作用将人类 DNA 连接酶 IIIα 压缩在灵活的 DNA 修复复合物中

Michal Hammel, Ishtiaque Rashid, Aleksandr Sverzhinsky, Yasin Pourfarjam, Miaw-Sheue Tsai, Tom Ellenberger, John M Pascal, In-Kwon Kim, John A Tainer, Alan E Tomkinson

Androgen signaling uses a writer and a reader of ADP-ribosylation to regulate protein complex assembly

雄激素信号传导使用 ADP-核糖基化的写入器和读取器来调节蛋白质复合物的组装

Chun-Song Yang, Kasey Jividen, Teddy Kamata, Natalia Dworak, Luke Oostdyk, Bartlomiej Remlein, Yasin Pourfarjam, In-Kwon Kim, Kang-Ping Du, Tarek Abbas, Nicholas E Sherman, David Wotton, Bryce M Paschal

The effects of synthetic orally administrated insulin nanoparticles in comparison to injectable insulin on the renal function markers of type 1- diabetic rats

合成口服胰岛素纳米颗粒与注射胰岛素对1型糖尿病大鼠肾功能指标的影响比较

Kheiripour, Nejat; Alipoor, Behnam; Ranjbar, Akram; Pourfarjam, Yasin; Kazemi Najafabadi, Farzaneh; Dehkhodaei, Narges; Farhadiannezhad, Masoumeh; Ghasemi, Hassan

Selective small molecule PARG inhibitor causes replication fork stalling and cancer cell death

选择性小分子 PARG 抑制剂导致复制叉停滞和癌细胞死亡

Jerry H Houl, Zu Ye, Chris A Brosey, Lakshitha P F Balapiti-Modarage, Sarita Namjoshi, Albino Bacolla, Daniel Laverty, Brian L Walker, Yasin Pourfarjam, Leslie S Warden, Naga Babu Chinnam, Davide Moiani, Roderick A Stegeman, Mei-Kuang Chen, Mien-Chie Hung, Zachary D Nagel, Tom Ellenberger, In-Kwon K

Effect of Cichorium intybus L. seed extract on renal parameters in experimentally induced early and late diabetes type 2 in rats

菊苣种子提取物对实验诱导的2型糖尿病早期和晚期大鼠肾脏参数的影响

Pourfarjam, Yasin; Rezagholizadeh, Lotfollah; Nowrouzi, Azin; Meysamie, Alipasha; Ghaseminejad, Sarah; Ziamajidi, Nasrin; Norouzi, Davood

Effect of Cichorium intybus L. on the expression of hepatic NF-κB and IKKβ and serum TNF-α in STZ- and STZ+ niacinamide-induced diabetes in rats

菊苣对STZ和STZ+烟酰胺诱发的糖尿病大鼠肝脏NF-κB和IKKβ表达及血清TNF-α的影响

Lotfollah Rezagholizadeh, Yasin Pourfarjam, Azin Nowrouzi, Manuchehr Nakhjavani, Alipasha Meysamie, Nasrin Ziamajidi, Peyman S Nowrouzi