日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A cryptic pocket in CB1 drives peripheral and functional selectivity

CB1 中的一个隐蔽口袋驱动外周和功能选择性

Rangari, Vipin Ashok; O'Brien, Evan S; Powers, Alexander S; Slivicki, Richard A; Bertels, Zachariah; Appourchaux, Kevin; Aydin, Deniz; Ramos-Gonzalez, Nokomis; Mwirigi, Juliet; Lin, Li; Mangutov, Elizaveta; Sobecks, Briana L; Awad-Agbaria, Yaseen; Uphade, Manoj B; Aguilar, Jhoan; Peddada, Teja Nikhil; Shiimura, Yuki; Huang, Xi-Ping; Folarin-Hines, Jakayla; Payne, Maria; Kalathil, Anirudh; Varga, Balazs R; Kobilka, Brian K; Pradhan, Amynah A; Cameron, Michael D; Kumar, Kaavya Krishna; Dror, Ron O; Gereau, Robert W 4th; Majumdar, Susruta

Structure-guided design of partial agonists at an opioid receptor.

基于结构的阿片受体部分激动剂设计

Varga Balazs R, Bernhard Sarah M, El Daibani Amal, Zaidi Saheem A, Lam Jordy H, Aguilar Jhoan, Appourchaux Kevin, Nazarova Antonina L, Kouvelis Alexa, Shinouchi Ryosuke, Hammond Haylee R, Eans Shainnel O, Weinreb Violetta, Margolis Elyssa B, Fay Jonathan F, Huang Xi-Ping, Pradhan Amynah, Katritch Vsevolod, McLaughlin Jay P, Majumdar Susruta, Che Tao

Enhancement of the endocannabinoid system through monoacylglycerol lipase inhibition relieves migraine-associated pain in mice

通过抑制单酰甘油脂肪酶增强内源性大麻素系统可缓解小鼠偏头痛相关疼痛

Mangutov, Elizaveta; Awad-Igbaria, Yaseen; Siegersma, Kendra; Gastambide, Francois; Asuni, Ayodeji A; Pradhan, Amynah A A

Activation of δ-opioid receptors blocks allodynia in a model of headache induced by PACAP

δ-阿片受体的激活可阻断PACAP诱导的头痛模型中的痛觉过敏。

Mangutov, Elizaveta; Dripps, Isaac; Siegersma, Kendra; Zhang, Yanping; Bocian, Rebecca; Asif, Sarah; Halbesma, Timothy; Witkowski, Wiktor; Pradhan, Amynah A

Delta opioid receptors: Overlooked outlier or the next big thing

δ阿片受体:被忽视的异类还是下一个重大发现

El Daibani, Amal; Burgess, Gwendolyn; Rysztak, Lauren; Jutkiewicz, Emily; Pradhan, Amynah A

Combination Targeted Therapy in Relapsed Diffuse Large B-Cell Lymphoma

复发性弥漫性大B细胞淋巴瘤的联合靶向治疗

Melani, Christopher; Lakhotia, Rahul; Pittaluga, Stefania; Phelan, James D; Huang, Da Wei; Wright, George; Simard, Jillian; Muppidi, Jagan; Thomas, Craig J; Ceribelli, Michele; Tosto, Frances A; Yang, Yandan; Xu, Weihong; Davies-Hill, Theresa; Pack, Svetlana D; Peer, Cody J; Arisa, Oluwatobi; Mena, Esther; Lindenberg, Liza; Bergvall, Ethan; Portell, Craig A; Farah, Rafic J; Lee, Seung Tae; Pradhan, Amynah; Morrison, Candis; Tadese, Atekelt; Juanitez, Anna Marie; Lu, Crystal; Jacob, Allison; Simmons, Heidi; Figg, William D; Steinberg, Seth M; Jaffe, Elaine S; Roschewski, Mark; Staudt, Louis M; Wilson, Wyndham H

Glial activation in pain and emotional processing regions in the nitroglycerin mouse model of chronic migraine

硝酸甘油诱导慢性偏头痛小鼠模型中疼痛和情绪处理区域的神经胶质细胞激活

Cropper, Haley C; Conway, Catherine M; Wyche, Whitney; Pradhan, Amynah A

Identification of 1,3,8-Triazaspiro[4.5]Decane-2,4-Dione Derivatives as a Novel δ Opioid Receptor-Selective Agonist Chemotype

鉴定出1,3,8-三氮杂螺[4.5]癸烷-2,4-二酮衍生物为一种新型δ阿片受体选择性激动剂化学型

Meqbil, Yazan J; Aguilar, Jhoan; Blaine, Arryn T; Chen, Lan; Cassell, Robert J; Pradhan, Amynah A; van Rijn, Richard M

A non-convulsant delta-opioid receptor agonist, KNT-127, reduces cortical spreading depression and nitroglycerin-induced allodynia

一种非惊厥性δ-阿片受体激动剂KNT-127可减轻皮质扩散性抑制和硝酸甘油诱导的痛觉过敏。

Bertels, Zachariah; Witkowski, Wiktor D; Asif, Sarah; Siegersma, Kendra; van Rijn, Richard M; Pradhan, Amynah A

Alternative Splicing Mechanisms Underlying Opioid-Induced Hyperalgesia

阿片类药物诱导痛觉过敏的替代剪接机制

Zhang, Pan; Perez, Olivia C; Southey, Bruce R; Sweedler, Jonathan V; Pradhan, Amynah A; Rodriguez-Zas, Sandra L