日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A mechanistically novel peptide agonist of the IL-7 receptor that addresses limitations of IL-7 cytokine therapy

一种机制新颖的 IL-7 受体肽激动剂,可解决 IL-7 细胞因子治疗的局限性

William J Dower, Angie Inkyung Park, Alice V Bakker, Steven E Cwirla, Praechompoo Pongtornpipat, Blake M Williams, Prarthana Joshi, Bryan A Baxter, Michael C Needels, Ronald W Barrett

Target-Based Screening against eIF4A1 Reveals the Marine Natural Product Elatol as a Novel Inhibitor of Translation Initiation with In Vivo Antitumor Activity

针对 eIF4A1 的靶向筛选表明,海洋天然产物 Elatol 是一种具有体内抗肿瘤活性的新型翻译起始抑制剂

Tara L Peters, Joseph Tillotson, Alison M Yeomans, Sarah Wilmore, Elizabeth Lemm, Carlos Jiménez-Romero, Luis A Amador, Lingxiao Li, Amit D Amin, Praechompoo Pongtornpipat, Christopher J Zerio, Andrew J Ambrose, Gillian Paine-Murrieta, Patricia Greninger, Francisco Vega, Cyril H Benes, Graham Packha

TKI sensitivity patterns of novel kinase-domain mutations suggest therapeutic opportunities for patients with resistant ALK+ tumors

新型激酶结构域突变的 TKI 敏感性模式为耐药 ALK+ 肿瘤患者提供了治疗机会

Amit Dipak Amin, Lingxiao Li, Soumya S Rajan, Vijay Gokhale, Matthew J Groysman, Praechompoo Pongtornpipat, Edgar O Tapia, Mengdie Wang, Jonathan H Schatz

Control of translational activation by PIM kinase in activated B-cell diffuse large B-cell lymphoma confers sensitivity to inhibition by PIM447

在活化的 B 细胞弥漫性大 B 细胞淋巴瘤中,PIM 激酶对翻译激活的控制赋予了对 PIM447 抑制的敏感性

Tara L Peters, Lingxiao Li, Ana A Tula-Sanchez, Praechompoo Pongtornpipat, Jonathan H Schatz

Evidence Suggesting That Discontinuous Dosing of ALK Kinase Inhibitors May Prolong Control of ALK+ Tumors

有证据表明,间断服用 ALK 激酶抑制剂可能会延长对 ALK+ 肿瘤的控制时间

Amit Dipak Amin, Soumya S Rajan, Winnie S Liang, Praechompoo Pongtornpipat, Matthew J Groysman, Edgar O Tapia, Tara L Peters, Lori Cuyugan, Jonathan Adkins, Lisa M Rimsza, Yves A Lussier, Soham D Puvvada, Jonathan H Schatz