日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dopamine D1 receptor activation in the striatum is sufficient to drive reinforcement of anteceding cortical patterns

纹状体中多巴胺D1受体的激活足以驱动先前皮层模式的强化。

Nuria Vendrell-Llopis ,Jonathan Read ,Samantha Boggiano ,Belinda Hetzler ,Zisis Peitsinis ,Cherise Stanley ,Meike Visel ,Dirk Trauner ,Prashant Donthamsetti ,Jose Carmena ,Stephan Lammel ,Ehud Y Isacoff

In-Cell Arrestin-Receptor Interaction Assays

细胞内 Arrestin 受体相互作用试验

Chen Zheng, Jonathan A Javitch, Nevin A Lambert, Prashant Donthamsetti, Vsevolod V Gurevich

Arrestin recruitment to dopamine D2 receptor mediates locomotion but not incentive motivation

Arrestin 募集到多巴胺 D2 受体介导运动但不介导激励动机

Prashant Donthamsetti #, Eduardo F Gallo #, David C Buck, Edward L Stahl, Ying Zhu, J Robert Lane, Laura M Bohn, Kim A Neve, Christoph Kellendonk, Jonathan A Javitch

Regional Heterogeneity of D2-Receptor Signaling in the Dorsal Striatum and Nucleus Accumbens

背侧纹状体和伏隔核中 D2 受体信号的区域异质性

Pamela F Marcott, Sheng Gong, Prashant Donthamsetti, Steven G Grinnell, Melissa N Nelson, Amy H Newman, Lutz Birnbaumer, Kirill A Martemyanov, Jonathan A Javitch, Christopher P Ford

Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D3 Receptor

了解多巴胺 D3 受体部分激动的结构基础

Mayako Michino, Comfort A Boateng, Prashant Donthamsetti, Hideaki Yano, Oluyomi M Bakare, Alessandro Bonifazi, Michael P Ellenberger, Thomas M Keck, Vivek Kumar, Clare Zhu, Ravi Verma, Jeffrey R Deschamps, Jonathan A Javitch, Amy Hauck Newman, Lei Shi

The role of kinetic context in apparent biased agonism at GPCRs

动力学背景在 GPCR 表观偏向激动中的作用

Carmen Klein Herenbrink, David A Sykes, Prashant Donthamsetti, Meritxell Canals, Thomas Coudrat, Jeremy Shonberg, Peter J Scammells, Ben Capuano, Patrick M Sexton, Steven J Charlton, Jonathan A Javitch, Arthur Christopoulos, J Robert Lane

Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity

(R)-5-(甲氨基)-5,6-二氢-4H-咪唑并[4,5,1-ij]喹啉-2(1H)-酮(Sumanirole)的新型类似物为多巴胺 D2/D3 受体激动剂的选择性提供线索

Mu-Fa Zou, Thomas M Keck, Vivek Kumar, Prashant Donthamsetti, Mayako Michino, Caitlin Burzynski, Catherine Schweppe, Alessandro Bonifazi, R Benjamin Free, David R Sibley, Aaron Janowsky, Lei Shi, Jonathan A Javitch, Amy Hauck Newman

Development of a Rapid Insulin Assay by Homogenous Time-Resolved Fluorescence

通过均相时间分辨荧光开发快速胰岛素检测方法

Zachary J Farino, Travis J Morgenstern, Julie Vallaghe, Nathalie Gregor, Prashant Donthamsetti, Paul E Harris, Nicolas Pierre, Robin Freyberg, Fabienne Charrier-Savournin, Jonathan A Javitch, Zachary Freyberg

Using Bioluminescence Resonance Energy Transfer (BRET) to Characterize Agonist-Induced Arrestin Recruitment to Modified and Unmodified G Protein-Coupled Receptors

使用生物发光共振能量转移 (BRET) 来表征激动剂诱导的 Arrestin 对修饰和未修饰的 G 蛋白偶联受体的募集

Prashant Donthamsetti, Jose Rafael Quejada, Jonathan A Javitch, Vsevolod V Gurevich, Nevin A Lambert

A new mechanism of allostery in a G protein-coupled receptor dimer

蛋白偶联受体二聚体的变构新机制

J Robert Lane, Prashant Donthamsetti, Jeremy Shonberg, Christopher J Draper-Joyce, Samuel Dentry, Mayako Michino, Lei Shi, Laura López, Peter J Scammells, Ben Capuano, Patrick M Sexton, Jonathan A Javitch, Arthur Christopoulos