日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into MERS and SARS coronavirus membrane proteins

对中东呼吸综合征(MERS)和严重急性呼吸综合征(SARS)冠状病毒膜蛋白的结构解析

Mann, Mandeep Kaur; Yin, Yanting; Marsili, Simone; Xie, Jiexiong; Doijen, Jordi; Miller, Robyn; Piassek, Madison; van den Broeck, Nick; Kariuki, Christopher Kinyanjui; de Gruyter, Heidi L M; Leijs, Anouk A; Snijder, Eric J; van Hemert, Martijn J; Keustermans, Ken; Van Gool, Michiel; Yu, Xiaodi; Loock, Marnix van; Koul, Anil; Sharma, Sujata; Van Damme, Ellen; Abeywickrema, Pravien

Discovery of a non-nucleoside inhibitor that binds to a novel site in the palm domain of the respiratory syncytial virus RNA-dependent RNA polymerase.

发现一种非核苷类抑制剂,可与呼吸道合胞病毒 RNA 依赖性 RNA 聚合酶掌状结构域中的新位点结合

Kalin Jay H, Yin Yanting, Tran Minh T, Piassek Madison, Fung Amy, Grosse Sandrine, Jacoby Edgar, Bhaumik Anusarka, Adhikary Suraj, Miller Robyn, Lemmens Cynthia, Lutter Ferdinand H, Pieters Serge, Cooymans Ludwig, Rombouts Geert, Oehlrich Daniel, Tomaso Sonia, Lozada Kate, Garcia Miguel Osorio, Anson Brandon, De Bruyn Suzanne, Smith-Monroy Constance, Neefs Jean-Marc, Conceição-Neto Nádia, Stoops Bart, van Vlijmen Herman, Patrick Aaron, Yu Xiaodi, Wong Victoria, Krosky Daniel, Abeywickrema Pravien, Mason Stephen, Jin Zhinan, Jonckers Tim H M, Sharma Sujata

Cannabidiol Toxicity Driven by Hydroxyquinone Formation

羟醌形成导致的大麻二酚毒性

Metzli I Montero, Pravien S Rajaram, Jose E Zamora Alvarado, Kara E McCloskey, Ryan D Baxter, Roberto C Andresen Eguiluz

High-Throughput Assessment of Bile Salt Export Pump Inhibition Using RapidFire-MS and DESI-MS

利用 RapidFire-MS 和 DESI-MS 对胆汁酸输出泵抑制进行高通量评估

Li, Jie; Morato, Nicolás M; Westover, Lori S; Abeywickrema, Pravien; Geng, Jieping; Piassek, Madison; Harden, David; Strambeanu, Iulia; Shi, Zhicai; Cooks, R Graham; Meng, Juncai

Engineering a cleaved, prefusion-stabilized influenza B virus hemagglutinin by identification and locking of all six pH switches

通过识别和锁定所有六个 pH 开关来设计裂解的、融合前稳定的乙型流感病毒血凝素

Jarek Juraszek, Fin J Milder, Xiaodi Yu, Sven Blokland, Daan van Overveld, Pravien Abeywickrema, Sem Tamara, Sujata Sharma, Lucy Rutten, Mark J G Bakkers, Johannes P M Langedijk

Convergence of immune escape strategies highlights plasticity of SARS-CoV-2 spike

免疫逃逸策略的融合凸显了 SARS-CoV-2 刺突蛋白的可塑性

Xiaodi Yu, Jarek Juraszek, Lucy Rutten, Mark J G Bakkers, Sven Blokland, Jelle M Melchers, Niels J F van den Broek, Annemiek Y W Verwilligen, Pravien Abeywickrema, Johan Vingerhoets, Jean-Marc Neefs, Shah A Mohamed Bakhash, Pavitra Roychoudhury, Alex Greninger, Sujata Sharma, Johannes P M Langedijk

Structural and mechanistic insights into the inhibition of respiratory syncytial virus polymerase by a non-nucleoside inhibitor

非核苷抑制剂抑制呼吸道合胞病毒聚合酶的结构和机制见解

Xiaodi Yu #, Pravien Abeywickrema #, Brecht Bonneux, Ishani Behera, Brandon Anson, Edgar Jacoby, Amy Fung, Suraj Adhikary, Anusarka Bhaumik, Rodrigo J Carbajo, Suzanne De Bruyn, Robyn Miller, Aaron Patrick, Quyen Pham, Madison Piassek, Nick Verheyen, Afzaal Shareef, Priscila Sutto-Ortiz, Nina Ysebae

Structural understanding of non-nucleoside inhibition in an elongating herpesvirus polymerase.

对延伸疱疹病毒聚合酶中非核苷类抑制剂的结构理解

Hayes Robert P, Heo Mee Ra, Mason Mark, Reid John, Burlein Christine, Armacost Kira A, Tellers David M, Raheem Izzat, Shaw Anthony W, Murray Edward, McKenna Philip M, Abeywickrema Pravien, Sharma Sujata, Soisson Stephen M, Klein Daniel

The methyltransferase domain of the Respiratory Syncytial Virus L protein catalyzes cap N7 and 2'-O-methylation

呼吸道合胞病毒L蛋白的甲基转移酶结构域催化N7帽和2'-O-甲基化。

Sutto-Ortiz, Priscila; Tcherniuk, Sergey; Ysebaert, Nina; Abeywickrema, Pravien; Noël, Mathieu; Decombe, Alice; Debart, Françoise; Vasseur, Jean-Jacques; Canard, Bruno; Roymans, Dirk; Rigaux, Peter; Eléouët, Jean-François; Decroly, Etienne

Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

氨基甲酸酯和N-嘧啶可减轻酰胺水解:基于结构的四氢喹啉IDO1抑制剂药物设计

Li, Derun; Deng, Yongqi; Achab, Abdelghani; Bharathan, Indu; Hopkins, Brett Andrew; Yu, Wensheng; Zhang, Hongjun; Sanyal, Sulagna; Pu, Qinglin; Zhou, Hua; Liu, Kun; Lim, Jongwon; Fradera, Xavier; Lesburg, Charles A; Lammens, Alfred; Martinot, Theodore A; Cohen, Ryan D; Doty, Amy C; Ferguson, Heidi; Nickbarg, Elliott B; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Abeywickrema, Pravien; Andrews, Christine; Chamberlin, Chad; Mabrouk, Omar; Curran, Patrick; Richards, Matthew; Saradjian, Peter; Miller, J Richard; Knemeyer, Ian; Otte, Karin M; Vincent, Stella; Sciammetta, Nunzio; Pasternak, Alexander; Bennett, David Jonathan; Han, Yongxin