日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibition of BET Bromodomain Proteins with GS-5829 and GS-626510 in Uterine Serous Carcinoma, a Biologically Aggressive Variant of Endometrial Cancer

使用 GS-5829 和 GS-626510 抑制子宫浆液性癌(一种生物侵袭性子宫内膜癌变体)中的 BET 溴结构域蛋白

Elena Bonazzoli, Federica Predolini, Emiliano Cocco, Stefania Bellone, Gary Altwerger, Gulden Menderes, Luca Zammataro, Anna Bianchi, Francesca Pettinella, Francesco Riccio, Chanhee Han, Ghanshyam Yadav, Salvatore Lopez, Aranzazu Manzano, Paola Manara, Natalia Buza, Pei Hui, Serena Wong, Babak Litko

SYD985, a Novel Duocarmycin-Based HER2-Targeting Antibody-Drug Conjugate, Shows Antitumor Activity in Uterine and Ovarian Carcinosarcoma with HER2/Neu Expression

SYD985 是一种新型的基于双卡霉素的靶向 HER2 的抗体药物偶联物,在表达 HER2/Neu 的子宫癌和卵巢癌肉瘤中显示出抗肿瘤活性。

Menderes, Gulden; Bonazzoli, Elena; Bellone, Stefania; Black, Jonathan; Predolini, Federica; Pettinella, Francesca; Masserdotti, Alice; Zammataro, Luca; Altwerger, Gary; Buza, Natalia; Hui, Pei; Wong, Serena; Litkouhi, Babak; Ratner, Elena; Silasi, Dan-Arin; Azodi, Masoud; Schwartz, Peter E; Santin, Alessandro D

Dual-Targeting Nanoparticles for In Vivo Delivery of Suicide Genes to Chemotherapy-Resistant Ovarian Cancer Cells

用于体内递送自杀基因至化疗耐药卵巢癌细胞的双靶向纳米颗粒

Cocco, Emiliano; Deng, Yang; Shapiro, Erik M; Bortolomai, Ileana; Lopez, Salvatore; Lin, Ken; Bellone, Stefania; Cui, Jiajia; Menderes, Gulden; Black, Jonathan D; Schwab, Carlton L; Bonazzoli, Elena; Yang, Fan; Predolini, Federica; Zammataro, Luca; Altwerger, Gary; de Haydu, Christopher; Clark, Mitchell; Alvarenga, Julio; Ratner, Elena; Azodi, Masoud; Silasi, Dan-Arin; Schwartz, Peter E; Litkouhi, Babak; Saltzman, W Mark; Santin, Alessandro D

Polymerase ε (POLE) ultra-mutation in uterine tumors correlates with T lymphocyte infiltration and increased resistance to platinum-based chemotherapy in vitro

子宫肿瘤中的聚合酶ε(POLE)超突变与 T 淋巴细胞浸润和体外对铂类化疗的耐药性增加相关

Stefania Bellone, Eliana Bignotti, Silvia Lonardi, Francesca Ferrari, Floriana Centritto, Alice Masserdotti, Francesca Pettinella, Jonathan Black, Gulden Menderes, Gary Altwerger, Pei Hui, Salvatore Lopez, Christopher de Haydu, Elena Bonazzoli, Federica Predolini, Luca Zammataro, Emiliano Cocco, Fed

Solitomab, an EpCAM/CD3 bispecific antibody construct (BiTE), is highly active against primary uterine serous papillary carcinoma cell lines in vitro

Solitomab是一种EpCAM/CD3双特异性抗体构建体(BiTE),在体外对原发性子宫浆液性乳头状癌细胞系具有很高的活性。

Bellone, Stefania; Black, Jonathan; English, Diana P; Schwab, Carlton L; Lopez, Salvatore; Cocco, Emiliano; Bonazzoli, Elena; Predolini, Federica; Ferrari, Francesca; Ratner, Elena; Silasi, Dan-Arin; Azodi, Masoud; Schwartz, Peter E; Santin, Alessandro D

Dual CCNE1/PIK3CA targeting is synergistic in CCNE1-amplified/PIK3CA-mutated uterine serous carcinomas in vitro and in vivo

CCNE1/PIK3CA 双靶向作用在体外和体内 CCNE1 扩增/PIK3CA 突变的子宫浆液性癌中具有协同作用

Emiliano Cocco, Salvatore Lopez, Jonathan Black, Stefania Bellone, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Carlton L Schwab, Gulden Menderes, Luca Zammataro, Natalia Buza, Pei Hui, Serena Wong, Siming Zhao, Yalai Bai, David L Rimm, Elena Ratner, Babak Litkouhi, Dan-Arin Silasi, Masou

Mutational landscape of uterine and ovarian carcinosarcomas implicates histone genes in epithelial-mesenchymal transition

子宫和卵巢癌肉瘤的突变图谱表明组蛋白基因参与了上皮-间质转化

Siming Zhao, Stefania Bellone, Salvatore Lopez, Durga Thakral, Carlton Schwab, Diana P English, Jonathan Black, Emiliano Cocco, Jungmin Choi, Luca Zammataro, Federica Predolini, Elena Bonazzoli, Mark Bi, Natalia Buza, Pei Hui, Serena Wong, Maysa Abu-Khalaf, Antonella Ravaggi, Eliana Bignotti, Elisab

Solitomab, an EpCAM/CD3 bispecific antibody construct (BiTE®), is highly active against primary uterine and ovarian carcinosarcoma cell lines in vitro

Solitomab 是一种 EpCAM/CD3 双特异性抗体构建体 (BiTE®),在体外对原发性子宫癌和卵巢癌肉瘤细胞系具有很高的活性。

Ferrari, Francesca; Bellone, Stefania; Black, Jonathan; Schwab, Carlton L; Lopez, Salvatore; Cocco, Emiliano; Bonazzoli, Elena; Predolini, Federica; Menderes, Gulden; Litkouhi, Babak; Ratner, Elena; Silasi, Dan-Arin; Azodi, Masoud; Schwartz, Peter E; Santin, Alessandro D

PIK3CA oncogenic mutations represent a major mechanism of resistance to trastuzumab in HER2/neu overexpressing uterine serous carcinomas

PIK3CA 致癌突变是 HER2/neu 过度表达的子宫浆液性癌对曲妥珠单抗产生耐药性的主要机制

Jonathan D Black, Salvatore Lopez, Emiliano Cocco, Stefania Bellone, Gary Altwerger, Carlton L Schwab, Diana P English, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Peter E Schwartz, Alessandro D Santin

Dual HER2/PIK3CA Targeting Overcomes Single-Agent Acquired Resistance in HER2-Amplified Uterine Serous Carcinoma Cell Lines In Vitro and In Vivo

HER2/PIK3CA 双靶向治疗在体内和体外克服了 HER2 扩增子宫浆液性癌细胞系中单药获得性耐药性

Salvatore Lopez, Emiliano Cocco, Jonathan Black, Stefania Bellone, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Carlton L Schwab, Diana P English, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Peter E Schwartz, Corrado Terranova, Roberto Angioli, Alessandro D Santin