日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Stereoselective Bio-Organocatalytic Cascade to Chiral Amides as Active Pharmaceutical Ingredient Intermediates Using ω-Transaminase and Choline Chloride Under Microwave Irradiation

利用ω-转氨酶和氯化胆碱在微波辐射下进行立体选择性生物有机催化级联反应,合成手性酰胺作为活性药物成分中间体

Romano, Salvatore; Damian, Matteo; Nardi, Monica; Procopio, Antonio; Strähler, Sebastian; Preschel, Daniël; Oliverio, Manuela; Mutti, Francesco G

Iron-Catalysed Carbene Transfer to Isocyanides as a Platform for Heterocycle Synthesis

铁催化卡宾向异氰化物转移作为杂环合成平台

Roose, Thomas R; Preschel, H Daniel; Mayo Tejedor, Helena; Roozee, Jasper C; Hamlin, Trevor A; Maes, Bert U W; Ruijter, Eelco; Orru, Romano V A

Multicomponent Synthesis of the SARS-CoV-2 Main Protease Inhibitor Nirmatrelvir

SARS-CoV-2 主要蛋白酶抑制剂 Nirmatrelvir 的多组分合成

H Daniel Preschel, Ruben T Otte, Ying Zhuo, Rebecca E Ruscoe, Ashleigh J Burke, Rachel Kellerhals, Brendan Horst, Sven Hennig, Elwin Janssen, Anthony P Green, Nicholas J Turner, Eelco Ruijter