日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and PET Imaging Biodistribution Studies of Radiolabeled Iododiflunisal, a Transthyretin Tetramer Stabilizer, Candidate Drug for Alzheimer's Disease

放射性标记的碘二氟尼柳(一种转甲状腺素四聚体稳定剂,阿尔茨海默病候选药物)的合成及PET成像生物分布研究

Joshi, Sameer M; Wilson, Thomas C; Li, Zibo; Preshlock, Sean; Gómez-Vallejo, Vanessa; Gouverneur, Véronique; Llop, Jordi; Arsequell, Gemma

Tandem Iridium-Catalyzed C-H Borylation/Copper-Mediated Radiofluorination of Aromatic C-H Bonds with [(18)F]TBAF

串联铱催化CH硼化/铜介导芳香族CH键放射性氟化反应(使用[(18)F]TBAF)

Morales, Maria; Preshlock, Sean; Sharninghausen, Liam S; Wright, Jay S; Brooks, Allen F; Sanford, Melanie S; Scott, Peter J H

Strategies for the Production of [11C]LY2795050 for Clinical Use

临床用[11C]LY2795050的生产策略

Tanpreet Kaur, Xia Shao, Mami Horikawa, Liam S Sharninghausen, Sean Preshlock, Allen F Brooks, Bradford D Henderson, Robert A Koeppe, Alexandre F DaSilva, Melanie S Sanford, Peter J H Scott

Copper-Mediated Radiocyanation of Unprotected Amino Acids and Peptides

铜介导的未保护氨基酸和肽的放射性氰化反应

Sharninghausen, Liam S; Preshlock, Sean; Joy, Stephen T; Horikawa, Mami; Shao, Xia; Winton, Wade P; Stauff, Jenelle; Kaur, Tanpreet; Koeppe, Robert A; Mapp, Anna K; Scott, Peter J H; Sanford, Melanie S

Sequential Ir/Cu-Mediated Method for the Meta-Selective C-H Radiofluorination of (Hetero)Arenes

用于(杂)芳烃间位选择性CH放射性氟化的顺序Ir/Cu介导方法

Wright, Jay S; Sharninghausen, Liam S; Preshlock, Sean; Brooks, Allen F; Sanford, Melanie S; Scott, Peter J H

Synthesis of Radiopharmaceuticals via "In-Loop" (11)C-Carbonylation as Exemplified by the Radiolabeling of Inhibitors of Bruton's Tyrosine Kinase

以布鲁顿酪氨酸激酶抑制剂的放射性标记为例,通过“环内”(11)C-羰基化合成放射性药物

Donnelly, David J; Preshlock, Sean; Kaur, Tanpreet; Tran, Tritin; Wilson, Thomas C; Mhanna, Karim; Henderson, Bradford D; Batalla, Daniel; Scott, Peter J H; Shao, Xia

Use of 55 PET radiotracers under approval of a Radioactive Drug Research Committee (RDRC)

经放射性药物研究委员会(RDRC)批准,使用55种PET放射性示踪剂

Jackson, Isaac M; Lee, So Jeong; Sowa, Alexandra R; Rodnick, Melissa E; Bruton, Laura; Clark, Mara; Preshlock, Sean; Rothley, Jill; Rogers, Virginia E; Botti, Leslie E; Henderson, Bradford D; Hockley, Brian G; Torres, Jovany; Raffel, David M; Brooks, Allen F; Frey, Kirk A; Kilbourn, Michael R; Koeppe, Robert A; Shao, Xia; Scott, Peter J H

Copper-Mediated Late-stage Radiofluorination: Five Years of Impact on Pre-clinical and Clinical PET Imaging

铜介导的后期放射性氟化:五年来对临床前和临床PET成像的影响

Wright, Jay S; Kaur, Tanpreet; Preshlock, Sean; Tanzey, Sean S; Winton, Wade P; Sharninghausen, Liam S; Wiesner, Nicholas; Brooks, Allen F; Sanford, Melanie S; Scott, Peter J H

Silyl phosphorus and nitrogen donor chelates for homogeneous ortho borylation catalysis

用于均相邻位硼化催化的硅基磷和氮供体螯合物

Ghaffari, Behnaz; Preshlock, Sean M; Plattner, Donald L; Staples, Richard J; Maligres, Peter E; Krska, Shane W; Maleczka, Robert E Jr; Smith, Milton R 3rd

A traceless directing group for C-H borylation

用于CH硼化的无痕导向基团

Preshlock, Sean M; Plattner, Donald L; Maligres, Peter E; Krska, Shane W; Maleczka, Robert E Jr; Smith, Milton R 3rd